The store will not work correctly when cookies are disabled.
JavaScript seems to be disabled in your browser. For the best experience on our site, be sure to turn on Javascript in your browser.
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 - ≥96%(HPLC), high purity , CAS No.208706-12-1
Potent and selective sst2agonist
Basic Description Synonyms N-[(1R)-2-[[[(1S*,3R*)-3-(Aminomethyl)cyclohexyl]methyl]amino]-1-(1H-indol-3-ylmethyl)-2-oxoethyl]spiro[1H-indene-1,4'-piperidine]-1'-carboxamide Specifications & Purity ≥96% Biochemical and Physiological Mechanisms Potent and selective somatostatin sst2receptor agonist (Kivalues are 4, 537, 2480, 3614 and 5017 nM for cloned human sst2, sst1, sst4, sst3and sst5receptors respectively). Storage Temp Store at 2-8°C Shipped In Wet ice
Names and Identifiers IUPAC Name N-[(2R)-1-[[(1R,3S)-3-(aminomethyl)cyclohexyl]methylamino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]spiro[indene-1,4'-piperidine]-1'-carboxamide INCHI InChI=1S/C33H41N5O2/c34-20-23-6-5-7-24(18-23)21-36-31(39)30(19-26-22-35-29-11-4-2-9-27(26)29)37-32(40)38-16-14-33(15-17-38)13-12-25-8-1-3-10-28(25)33/h1-4,8-13,22-24,30,35H,5-7,14-21,34H2,(H,36,39)(H,37,40)/t23-,24+,30+/m0/s1 InChi Key DAMXHAMKVXERLM-FVBCXUTKSA-N Canonical SMILES C1CC(CC(C1)CNC(=O)C(CC2=CNC3=CC=CC=C32)NC(=O)N4CCC5(CC4)C=CC6=CC=CC=C56)CN Isomeric SMILES C1C[C@@H](C[C@@H](C1)CNC(=O)[C@@H](CC2=CNC3=CC=CC=C32)NC(=O)N4CCC5(CC4)C=CC6=CC=CC=C56)CN PubChem CID 9915239 Molecular Weight 539.71
Chemical and Physical Properties Solubility Solvent:DMSO, Max Conc. mg/mL: 26.99, Max Conc. mM: 50; Solvent:ethanol, Max Conc. mg/mL: 53.97, Max Conc. mM: 100
Solution Calculators Molarity Calculator Determine the necessary mass, volume, or concentration for preparing a solution.
Dilution Calculator Determine the dilution needed to prepare a stock solution.
Reconstitution Calculator