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(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 - ≥96%(HPLC), high purity , CAS No.208706-12-1

  • ≥96%
Item Number
R287115
Grouped product items
SKUSizeAvailabilityPrice Qty
R287115-1mg
1mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$127.90
R287115-10mg
10mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$274.90

Potent and selective sst2agonist

Basic Description

SynonymsN-[(1R)-2-[[[(1S*,3R*)-3-(Aminomethyl)cyclohexyl]methyl]amino]-1-(1H-indol-3-ylmethyl)-2-oxoethyl]spiro[1H-indene-1,4'-piperidine]-1'-carboxamide
Specifications & Purity≥96%
Biochemical and Physiological MechanismsPotent and selective somatostatin sst2receptor agonist (Kivalues are 4, 537, 2480, 3614 and 5017 nM for cloned human sst2, sst1, sst4, sst3and sst5receptors respectively).
Storage TempStore at 2-8°C
Shipped InWet ice

Names and Identifiers

IUPAC Name N-[(2R)-1-[[(1R,3S)-3-(aminomethyl)cyclohexyl]methylamino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]spiro[indene-1,4'-piperidine]-1'-carboxamide
INCHI InChI=1S/C33H41N5O2/c34-20-23-6-5-7-24(18-23)21-36-31(39)30(19-26-22-35-29-11-4-2-9-27(26)29)37-32(40)38-16-14-33(15-17-38)13-12-25-8-1-3-10-28(25)33/h1-4,8-13,22-24,30,35H,5-7,14-21,34H2,(H,36,39)(H,37,40)/t23-,24+,30+/m0/s1
InChi Key DAMXHAMKVXERLM-FVBCXUTKSA-N
Canonical SMILES C1CC(CC(C1)CNC(=O)C(CC2=CNC3=CC=CC=C32)NC(=O)N4CCC5(CC4)C=CC6=CC=CC=C56)CN
Isomeric SMILES C1C[C@@H](C[C@@H](C1)CNC(=O)[C@@H](CC2=CNC3=CC=CC=C32)NC(=O)N4CCC5(CC4)C=CC6=CC=CC=C56)CN
PubChem CID 9915239
Molecular Weight 539.71

Certificates

Certificate of Analysis(COA)

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Chemical and Physical Properties

SolubilitySolvent:DMSO, Max Conc. mg/mL: 26.99, Max Conc. mM: 50; Solvent:ethanol, Max Conc. mg/mL: 53.97, Max Conc. mM: 100

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Solution Calculators