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AGC:Containing PKA, PKG, PKC families
4-[1-ethyl-7-(piperazin-1-ylmethyl)imidazo[4,5-c]pyridin-2-yl]-1,2,5-oxadiazol-3-amine , CAS No.E608979, Inhibitor of ribosomal protein S6 kinase A5

4-[1-ethyl-7-(piperazin-1-ylmethyl)imidazo[4,5-c]pyridin-2-yl]-1,2,5-oxadiazol-3-amine , CAS No.E608979, Inhibitor of ribosomal protein S6 kinase A5

Item Number

E608979

Grouped product items
SKU	Size	Availability	Price	Qty
E608979-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$600.90
E608979-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,000.90

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Basic Description

Synonyms	compound 24
Grade	Moligand™
Action Type	INHIBITOR
Mechanism of action	Inhibitor of ribosomal protein S6 kinase A5

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

IUPAC Name	4-[1-ethyl-7-(piperazin-1-ylmethyl)imidazo[4,5-c]pyridin-2-yl]-1,2,5-oxadiazol-3-amine
INCHI	InChI=1S/C15H20N8O/c1-2-23-13-10(9-22-5-3-17-4-6-22)7-18-8-11(13)19-15(23)12-14(16)21-24-20-12/h7-8,17H,2-6,9H2,1H3,(H2,16,21)
InChi Key	OXZLPOLYTISTQY-UHFFFAOYSA-N
Canonical SMILES	CCn1c(nc2c1c(CN1CCNCC1)cnc2)c1nonc1N
Isomeric SMILES	CCN1C2=C(C=NC=C2CN3CCNCC3)N=C1C4=NON=C4N
PubChem CID	44397277

ChEMBL Ligand	CHEMBL415770
PubChem CID	44397277

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1. Bamford MJ, Bailey N, Davies S, Dean DK, Francis L, Panchal TA, Parr CA, Sehmi S, Steadman JG, Takle AK et al.. (2005) (1H-imidazo[4,5-c]pyridin-2-yl)-1,2,5-oxadiazol-3-ylamine derivatives: further optimisation as highly potent and selective MSK-1-inhibitors.. Bioorg Med Chem Lett, 15 (14): (3407-11). [PMID:15955699]

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