5-[2-[5-[[4-[[4-(2-hydroxyethyl)piperazin-1-yl]methyl]-3-(trifluoromethyl)phenyl]carbamoyl]-2-methylphenyl]ethynyl]-N,1-dimethylimidazole-2-carboxamide , CAS No.H609459, Inhibitor of ABL proto-oncogene 1; non-receptor tyrosine kinase;Inhibitor of EPH receptor A2;Inhibitor of EPH receptor A3;Inhibitor of EPH receptor A7;Inhibitor of platelet derived growth factor receptor alpha;Inhibitor of ret proto-oncogene;Inhibitor of
5-[2-[5-[[4-[[4-(2-hydroxyethyl)piperazin-1-yl]methyl]-3-(trifluoromethyl)phenyl]carbamoyl]-2-methylphenyl]ethynyl]-N,1-dimethylimidazole-2-carboxamide , CAS No.H609459, Inhibitor of ABL proto-oncogene 1; non-receptor tyrosine kinase;Inhibitor of EPH receptor A2;Inhibitor of EPH receptor A3;Inhibitor of EPH receptor A7;Inhibitor of platelet derived growth factor receptor alpha;Inhibitor of ret proto-oncogene;Inhibitor of
Inhibitor of ABL proto-oncogene 1; non-receptor tyrosine kinase;Inhibitor of EPH receptor A2;Inhibitor of EPH receptor A3;Inhibitor of EPH receptor A7;Inhibitor of platelet derived growth factor receptor alpha;Inhibitor of ret proto-oncogene;Inhibitor of
1.Thomas M, Huang WS, Wen D, Zhu X, Wang Y, Metcalf CA, Liu S, Chen I, Romero J, Zou D et al.. (2011) Discovery of 5-(arenethynyl) hetero-monocyclic derivatives as potent inhibitors of BCR-ABL including the T315I gatekeeper mutant.. Bioorg Med Chem Lett, 21 (12):(3743-8). [PMID:21561767]
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