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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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I346768-1mg | 1mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $59.90 | |
I346768-5mg | 5mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $121.90 | |
I346768-10mg | 10mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $182.90 | |
I346768-25mg | 25mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $309.90 | |
I346768-50mg | 50mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $461.90 | |
I346768-100mg | 100mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $661.90 |
Synonyms | AM85665|J-014159|L-822179|UNII-1M7NI1A92L|.ALPHA. 5IA|3-(5-Methyl-1,2-oxazol-3-yl)-6-[(1-methyl-1H-1,2,3-triazol-4-yl)methoxy][1,2,4]triazolo[3,4-a]phthalazine|A14343|CS-0066094|5-methyl-3-[6-[(1-methyltriazol-4-yl)methoxy]-[1,2,4]triazolo[3,4-a]phthalazi |
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Specifications & Purity | Moligand™, ≥97% |
Storage Temp | Protected from light,Store at -20°C |
Shipped In | Ice chest + Ice pads |
Grade | Moligand™ |
Action Type | ALLOSTERIC MODULATOR |
Mechanism of action | Allosteric modulator of GABA A receptor α1 subunit;Allosteric modulator of GABA A receptor α2 subunit;Allosteric modulator of GABA A receptor α3 subunit;Allosteric modulator of GABA A receptor α5 subunit |
Product Description |
α5IA (L-822179) is a selective α5 GABAA receptor inverse agonist with neuroprotective potential.
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IUPAC Name | 5-methyl-3-[6-[(1-methyltriazol-4-yl)methoxy]-[1,2,4]triazolo[3,4-a]phthalazin-3-yl]-1,2-oxazole |
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INCHI | InChI=1S/C17H14N8O2/c1-10-7-14(22-27-10)16-20-19-15-12-5-3-4-6-13(12)17(21-25(15)16)26-9-11-8-24(2)23-18-11/h3-8H,9H2,1-2H3 |
InChi Key | NZMJFRXKGUCYNP-UHFFFAOYSA-N |
Canonical SMILES | CC1=CC(=NO1)C2=NN=C3N2N=C(C4=CC=CC=C43)OCC5=CN(N=N5)C |
Isomeric SMILES | CC1=CC(=NO1)C2=NN=C3N2N=C(C4=CC=CC=C43)OCC5=CN(N=N5)C |
Alternate CAS | 215874-86-5 |
PubChem CID | 6918451 |
MeSH Entry Terms | 3-(5-methylisoxazol-3-yl)-6-((1-methyl-1,2,3-triazol-4-yl)methyloxy)-1,2,4-triazolo(3,4-a)phthalazine;alpha5IA cpd |
Molecular Weight | 362.35 |
Enter Lot Number to search for COA:
To view the certificate results,please click on a Lot number.For Lot numbers from past orders,please use our order status section
Lot Number | Certificate Type | Date | Item |
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G2419102 | Certificate of Analysis | Apr 08, 2024 | I346768 |
G2419103 | Certificate of Analysis | Apr 08, 2024 | I346768 |
G2419112 | Certificate of Analysis | Apr 08, 2024 | I346768 |
G2419121 | Certificate of Analysis | Apr 08, 2024 | I346768 |
G2419122 | Certificate of Analysis | Apr 08, 2024 | I346768 |
G2419123 | Certificate of Analysis | Apr 08, 2024 | I346768 |
G2419124 | Certificate of Analysis | Apr 08, 2024 | I346768 |
G2419125 | Certificate of Analysis | Apr 08, 2024 | I346768 |
G2419126 | Certificate of Analysis | Apr 08, 2024 | I346768 |
G2419127 | Certificate of Analysis | Apr 08, 2024 | I346768 |
G2419128 | Certificate of Analysis | Apr 08, 2024 | I346768 |
G2419129 | Certificate of Analysis | Apr 08, 2024 | I346768 |
Solubility | Soluble in DMSO: >2 mg/mL |
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Sensitivity | light sensitive |