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AS 2034178 - ≥98%(HPLC), high purity , CAS No.1030846-42-4

Item Number

A288780

Grouped product items
SKU	Size	Availability	Price	Qty
A288780-10mg	10mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$206.90
A288780-50mg	50mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$808.90

Selective FFA1 (GPR40) agonist

Basic Description

Synonyms	2-Fluoro-4-[[[1,2,3,4-Tetrahydro-1-(2-phenoxyethyl)-5-quinolinyl]methyl]amino]benzenepropanoic acid
Specifications & Purity	≥98%(HPLC)
Biochemical and Physiological Mechanisms	Selective free fatty acid receptor 1 (FFA1/GPR40) agonist. Exhibits selectivity for GPR40 over GPR41, GPR43, GPR119, GPR120 and PPARγ. Induces glucose-dependent insulin secretion in pancreatic MIN6 cells andin vivo. Enhances insulin sensitivity in a type
Storage Temp	Store at 2-8°C
Shipped In	Wet ice

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

IUPAC Name	3-[2-fluoro-4-[[1-(2-phenoxyethyl)-3,4-dihydro-2H-quinolin-5-yl]methylamino]phenyl]propanoic acid
INCHI	InChI=1S/C27H29FN2O3/c28-25-18-22(13-11-20(25)12-14-27(31)32)29-19-21-6-4-10-26-24(21)9-5-15-30(26)16-17-33-23-7-2-1-3-8-23/h1-4,6-8,10-11,13,18,29H,5,9,12,14-17,19H2,(H,31,32)
InChi Key	VENOXIKBBUVHRY-UHFFFAOYSA-N
Canonical SMILES	C1CC2=C(C=CC=C2N(C1)CCOC3=CC=CC=C3)CNC4=CC(=C(C=C4)CCC(=O)O)F
Isomeric SMILES	C1CC2=C(C=CC=C2N(C1)CCOC3=CC=CC=C3)CNC4=CC(=C(C=C4)CCC(=O)O)F
PubChem CID	24808572
Molecular Weight	448.53

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Solubility	Solvent:DMSO, Max Conc. mg/mL: 22.43, Max Conc. mM: 50; Solvent:ethanol, Max Conc. mg/mL: 8.97, Max Conc. mM: 20

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