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Targets
G protein-coupled receptors (GPCRs)
Proteinase-activated receptors
AZ7188 - 95%, high purity , CAS No.A607845, Antagonist of PAR2

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AZ7188 - 95%, high purity , CAS No.A607845, Antagonist of PAR2

Moligand™
≥95%

Formula: C₁₇H₁₄N₂O
Molecular Weight: 262.31
PubChem CID: 129320516

Item Number

A607845

Grouped product items
SKU	Size	Availability	Price
A607845-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,000.90
A607845-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,000.90
A607845-100mg	100mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$5,602.90

View related series

Heterocyclic compound PAR2 Antagonist

Basic Description

Specifications & Purity	95%
Storage Temp	Store at 2-8°C
Shipped In	Wet ice
Grade	Moligand™
Action Type	ANTAGONIST
Mechanism of action	Antagonist of PAR2

Associated Targets

F2RL1 Tchem Proteinase-activated receptor 2 1 Activities

Discover Target: F2RL1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

IUPAC Name	2,3-dihydro-1'H-[2,3'-biindole]-1-carbaldehyde
INCHI	InChI=1S/C17H14N2O/c20-11-19-16-8-4-1-5-12(16)9-17(19)14-10-18-15-7-3-2-6-13(14)15/h1-8,10-11,17-18H,9H2
InChi Key	GFACBUCIUAKRSV-UHFFFAOYSA-N
Canonical SMILES	O=CN1c2ccccc2CC1c1c[nH]c2c1cccc2
PubChem CID	129320516
Molecular Weight	262.31

Database links

GPCRdb Ligand	AZ7188
PubChem CID	129320516

Certificates

Certificate of Analysis(COA)

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4 results found

Lot Number	Certificate Type	Date	Item
E2416143	Certificate of Analysis	Apr 28, 2024	A607845
E2416144	Certificate of Analysis	Apr 28, 2024	A607845
E2416145	Certificate of Analysis	Apr 28, 2024	A607845
E2416146	Certificate of Analysis	Apr 28, 2024	A607845

References

1. Cheng RKY, Fiez-Vandal C, Schlenker O, Edman K, Aggeler B, Brown DG, Brown GA, Cooke RM, Dumelin CE, Doré AS et al.. (2017) Structural insight into allosteric modulation of protease-activated receptor 2.. Nature, 545 (7652): (112-115). [PMID:28445455]

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