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BMS-962212 - 99%, high purity , CAS No.1430114-34-3

≥99%

CAS#: 1430114-34-3
Formula: C₃₂H₂₈ClFN₈O₅
Molecular Weight: 659.07
PubChem CID: 71548883

Item Number

B650175

Grouped product items
SKU	Size	Availability	Price
B650175-1mg	1mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$580.90
B650175-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,450.90
B650175-10mg	10mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,350.90

View related series

Factor Xa Metabolic Enzyme/Protease

Basic Description

Synonyms	BMS-962212\|1430114-34-3\|UNII-VWJ4VVZ3OU\|VWJ4VVZ3OU\|4-[[(1S)-2-[(E)-3-[3-chloro-2-fluoro-6-(tetrazol-1-yl)phenyl]prop-2-enoyl]-5-(4-methyl-2-oxopiperazin-1-yl)-3,4-dihydro-1H-isoquinoline-1-carbonyl]amino]benzoic acid\|(S,E)-4-(2-(3-(3-chloro-2-fluoro-6-(1h
Specifications & Purity	≥99%
Biochemical and Physiological Mechanisms	BMS-962212 is a direct, reversible, selective factor XIa (FXIa) inhibitor . BMS-962212 is well tolerated, with fast onset of pharmacodynamic (PD) responses and rapid elimination. BMS-962212 increases exposure dependently in activated partial thromboplasti
Storage Temp	Store at -20°C
Shipped In	Ice chest + Ice pads
Product Description	BMS-962212 is a direct, reversible, selective factor XIa (FXIa) inhibitor. BMS-962212 is well tolerated, with fast onset of pharmacodynamic (PD) responses and rapid elimination. BMS-962212 increases exposure dependently in activated partial thromboplastin time, and decreases exposure dependently in FXI clotting activity. Form:Solid

Associated Targets

F11 Tchem Coagulation factor XI 0 Activities

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F10 Tclin Coagulation factor X 0 Activities

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F9 Tchem Coagulation factor IX 0 Activities

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F12 Tchem Coagulation factor XII 0 Activities

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F7 Tchem Coagulation factor VII 0 Activities

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PROC Tchem Vitamin K-dependent protein C 0 Activities

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PLAT Tclin Tissue-type plasminogen activator 0 Activities

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PLG Tclin Plasminogen 0 Activities

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KLK1 Tchem Kallikrein-1 0 Activities

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KLKB1 Tclin Plasma kallikrein 0 Activities

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PLAU Tchem Urokinase-type plasminogen activator 0 Activities

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F2 Tclin Prothrombin 0 Activities

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Names and Identifiers

IUPAC Name	4-[[(1S)-2-[(E)-3-[3-chloro-2-fluoro-6-(tetrazol-1-yl)phenyl]prop-2-enoyl]-5-(4-methyl-2-oxopiperazin-1-yl)-3,4-dihydro-1H-isoquinoline-1-carbonyl]amino]benzoic acid
INCHI	InChI=1S/C32H28ClFN8O5/c1-39-15-16-40(28(44)17-39)25-4-2-3-22-21(25)13-14-41(30(22)31(45)36-20-7-5-19(6-8-20)32(46)47)27(43)12-9-23-26(42-18-35-37-38-42)11-10-24(33)29(23)34/h2-12,18,30H,13-17H2,1H3,(H,36,45)(H,46,47)/b12-9+/t30-/m0/s1
InChi Key	WYFCZWSWFGJODV-MIANJLSGSA-N
Canonical SMILES	CN1CCN(C(=O)C1)C2=CC=CC3=C2CCN(C3C(=O)NC4=CC=C(C=C4)C(=O)O)C(=O)C=CC5=C(C=CC(=C5F)Cl)N6C=NN=N6
Isomeric SMILES	CN1CCN(C(=O)C1)C2=CC=CC3=C2CCN([C@@H]3C(=O)NC4=CC=C(C=C4)C(=O)O)C(=O)/C=C/C5=C(C=CC(=C5F)Cl)N6C=NN=N6
Alternate CAS	1430114-34-3
PubChem CID	71548883
MeSH Entry Terms	4-(2-(3-(3-chloro-2-fluoro-6-(1H-tetrazol-1-yl)phenyl)acryloyl)-5-(4-methyl-2-oxopiperazin-1-yl)-1,2,3,4-tetrahydroisoquinoline-1-carboxamido)benzoic acid;BMS-962212
Molecular Weight	659.07

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