BP 897 is a potent and selective agonist of dopamine D3 receptor and a weak antagonist of dopamine D2 receptor with Ki of 0.92 nM and 61 nM for D3 and D2 receptors, respectively. BP 897 shows low affinities at D1 and D4 receptors with Ki of 3\u2009µM and
Storage Temp
Store at -20°C
Shipped In
Ice chest + Ice pads
Grade
Moligand™
Action Type
AGONIST
Mechanism of action
Agonist of D 3 receptor
Product Description
Information
BP 897 is a potent and selective agonist of dopamine D3 receptor and a weak antagonist of dopamine D2 receptor with Ki of 0.92 nM and 61 nM for D3 and D2 receptors, respectively. BP 897 shows low affinities at D1 and D4 receptors with Ki of 3 µM and 0.3 µM, respectively.
1.Pilla M, Perachon S, Sautel F, Garrido F, Mann A, Wermuth CG, Schwartz JC, Everitt BJ, Sokoloff P. (1999) Selective inhibition of cocaine-seeking behaviour by a partial dopamine D3 receptor agonist.. Nature, 400 (6742):(371-5). [PMID:10432116]
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F2429114