Determine the necessary mass, volume, or concentration for preparing a solution.
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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B608238-5mg | 5mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $700.90 | |
B608238-25mg | 25mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $2,000.90 |
Grade | Moligand™ |
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Action Type | CHANNEL BLOCKER |
Mechanism of action | Channel blocker of TRPC6 |
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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IUPAC Name | [2-(1,3-benzodioxol-5-ylamino)-1,3-thiazol-4-yl]-[(3R,5S)-3,5-dimethylpiperidin-1-yl]methanone |
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INCHI | InChI=1S/C18H21N3O3S/c1-11-5-12(2)8-21(7-11)17(22)14-9-25-18(20-14)19-13-3-4-15-16(6-13)24-10-23-15/h3-4,6,9,11-12H,5,7-8,10H2,1-2H3,(H,19,20)/t11-,12+ |
InChi Key | UBMOUBBRNPNZPM-TXEJJXNPSA-N |
Canonical SMILES | O1COC2=C1C=CC(=C2)NC=3SC=C(N3)C(=O)N4C[C@H](C[C@H](C4)C)C |
RCSB PDB Ligand | W99 |
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Enter Lot Number to search for COA:
1. Tang Q, Guo W, Zheng L, Wu JX, Liu M, Zhou X, Zhang X, Chen L. (2018) Structure of the receptor-activated human TRPC6 and TRPC3 ion channels.. Cell Res, 28 (7): (746-755). [PMID:29700422] |