Signal Transduction
Cancer is strongly associated with signal transduction changes. Our resources for cancer signal transduction include pathway cards covering cellular apoptosis, Akt, EGF, p53, VEGF and more.
- NG-Monomethyl-L-arginine Acetate
Specifications & Purity: ≥98%
CAS No.: 53308-83-1
Starting at $93.90
- SNAP [S-Nitroso-N-acetylpenicillamine]
Specifications & Purity: ≥97%
CAS No.: 67776-06-1
Starting at $24.90
- Ammonium pyrrolidinedithiocarbamate
Specifications & Purity: 99%
CAS No.: 5108-96-3
Starting at $9.90
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- 5-HT Receptor4item
- 5-HT1A receptor Agonist9item
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- 5-HT1B receptor Agonist7item
- 5-HT1B receptor Antagonist1 item
- 5-HT1D receptor Agonist6item
- 5-HT1D receptor Antagonist3item
- 5-ht1e receptor Agonist4item
- 5-HT1F receptor Agonist3item
- 5-HT2A receptor Agonist4item
- 5-HT2A receptor Antagonist16item
- 5-HT2B receptor Agonist3item
- 5-HT2B receptor Antagonist13item
- 5-HT2C receptor Agonist2item
- 5-HT2C receptor Antagonist12item
- 5-HT3A Antagonist5item
- 5-HT3AB Antagonist1 item
- 5-HT4 receptor Agonist1 item
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- A2B receptor Antagonist19item
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- ABL proto-oncogene 1,non-receptor tyrosine kinase Inhibitor1 item
- Accession#:P317492item
- Accession#:P317512item
- Accession#:P422262item
- Accession#:P607632item
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- Active ester1 item
- adenylyl cyclase 1 Inhibitor1 item
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- Ammonium transporter Rh type A1 item
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- BLT1 receptor Antagonist2item
- bromodomain containing 1 Inhibitor1 item
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- CaCC Channel blocker1 item
- Calcium Channel4item
- CaMK3item
- cancer research1 item
- carbonic anhydrase 1 Activator1 item
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- carbonic anhydrase 12 Inhibitor1 item
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- CaS receptor Allosteric modulator2item
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- CatSper1 Activator1 item
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- Cav1.1 Gating inhibitor2item
- Cav1.2 Gating inhibitor3item
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- CB1 receptor Agonist1 item
- CB1 receptor Antagonist6item
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- CB2 receptor Allosteric modulator1 item
- CB2 receptor Antagonist3item
- CCK1 receptor Agonist1 item
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- CCK2 receptor Agonist1 item
- CCK2 receptor Antagonist6item
- CCR43item
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- CCR3 Antagonist1 item
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- CCR5 Antagonist3item
- CCR8 Agonist1 item
- CDC like kinase 1 Inhibitor1 item
- CDC like kinase 3 Inhibitor1 item
- Cell Cycle/DNA Damage2item
- Cell signal transduction and Neuroscience2item
- CFTR Activator1 item
- checkpoint kinase 1 Inhibitor1 item
- checkpoint kinase 2 Inhibitor1 item
- Chelate / complex1 item
- chemerin receptor 1 Agonist1 item
- chemerin receptor 2 Agonist1 item
- Chemical Biology1 item
- CNGA1 Channel blocker1 item
- component of inhibitor of nuclear factor kappa B kinase complex Inhibitor1 item
- Constitutive androstane receptor Agonist1 item
- CoV 3C-like (main) protease Inhibitor1 item
- COX2item
- COX-2 Inhibitor1 item
- CRF1 receptor Antagonist2item
- CT receptor Agonist1 item
- Cx23 Inhibitor1 item
- Cx25 Inhibitor1 item
- Cx26 Inhibitor1 item
- Cx30 Inhibitor1 item
- Cx30.2 Inhibitor1 item
- Cx30.3 Inhibitor1 item
- Cx31 Inhibitor1 item
- Cx31.1 Inhibitor1 item
- Cx31.9 Inhibitor1 item
- Cx32 Inhibitor1 item
- Cx36 Inhibitor1 item
- Cx37 Inhibitor1 item
- Cx40 Inhibitor1 item
- Cx40.1 Inhibitor1 item
- Cx43 Inhibitor1 item
- Cx45 Inhibitor1 item
- Cx46 Inhibitor1 item
- Cx47 Inhibitor1 item
- cyclin dependent kinase 1 Inhibitor7item
- cyclin dependent kinase 2 Inhibitor5item
- cyclin dependent kinase 4 Inhibitor4item
- cyclin dependent kinase 5 Inhibitor5item
- cyclin dependent kinase 7 Inhibitor3item
- cyclin dependent kinase 9 Inhibitor2item
- Cyclopentadiene1 item
- CYP3A4 Inhibitor2item
- CysLT1 receptor Agonist2item
- CysLT1 receptor Antagonist2item
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- D1 receptor Agonist2item
- D2 receptor Agonist8item
- D2 receptor Antagonist11item
- D3 receptor Agonist6item
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- D4 receptor Agonist3item
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- Dopamine Receptor2item
- DP1 receptor Agonist2item
- DP1 receptor Antagonist4item
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- dual specificity tyrosine phosphorylation regulated kinase 1A Inhibitor2item
- Element classified compounds2item
- Endogenous Metabolite2item
- EP1 receptor Agonist2item
- EP1 receptor Antagonist4item
- EP2 receptor Agonist2item
- EP2 receptor Antagonist3item
- EP3 receptor Agonist2item
- EP3 receptor Antagonist3item
- EP4 receptor Agonist3item
- EP4 receptor Antagonist5item
- Epigenetics35item
- Estrogen receptor-α Agonist4item
- Estrogen receptor-β Agonist2item
- Estrogen receptor-β Antagonist3item
- ETA receptor Antagonist8item
- ETB receptor Antagonist3item
- ether1 item
- eukaryotic translation initiation factor 2 alpha kinase 2 Inhibitor2item
- FAAH4item
- FFA1 receptor Agonist4item
- FFA2 receptor Antagonist2item
- FFA4 receptor Agonist2item
- Five membered carbocyclic compound1 item
- Five-Membered Heterocyclic Compounds6item
- FL L-Cystine1 item
- Flavonoids1 item
- fms related receptor tyrosine kinase 3 Inhibitor2item
- FP receptor Agonist3item
- FPR2/ALX Agonist3item
- Functional group compounds3item
- furan1 item
- Fused ring tetrahydropyrans3item
- GABAA receptor α1 subunit Allosteric modulator2item
- GABAA receptor α2 subunit Allosteric modulator2item
- GABAA receptor α3 subunit Allosteric modulator2item
- GABAA receptor α5 subunit Allosteric modulator2item
- GABAA receptor α6 subunit Allosteric modulator2item
- GABAB receptor Agonist2item
- GABAB receptor Allosteric modulator2item
- GABAB receptor Antagonist4item
- GABAB1 Antagonist3item
- GAT1 Inhibitor2item
- Gene ID:100002item
- Gene ID:2072item
- Gene ID:2082item
- Gene ID:58812item
- Gene ID:67782item
- GLP-1 receptor Agonist3item
- GLP-2 receptor Agonist2item
- GluA1 Allosteric modulator2item
- GluA2 Allosteric modulator2item
- GluA3 Allosteric modulator2item
- GluA4 Allosteric modulator2item
- glucagon receptor Allosteric modulator2item
- Glucocorticoid receptor Agonist3item
- GluN1 Antagonist2item
- GluN2A Antagonist3item
- GluN2B Antagonist3item
- GluN2C Antagonist3item
- GluN2D Antagonist3item
- Glycine Receptor (All subtypes) Subunit-specific2item
- glycine receptor α2 subunit Antagonist2item
- glycogen synthase kinase 3 alpha Inhibitor2item
- glycogen synthase kinase 3 beta Inhibitor9item
- GnRH1 receptor Antagonist2item
- GPCR/G Protein55item
- GPR119 Agonist3item
- GPR17 Agonist2item
- GPR55 Agonist3item
- GPR55 Antagonist3item
- Guanylyl cyclase,α1β1 Activator2item
- H1 receptor Antagonist10item
- H2 receptor Antagonist4item
- H3 receptor Antagonist4item
- H4 receptor Antagonist4item
- Halogenated heterocyclic block1 item
- HCA2 receptor Agonist2item
- Histamine receptor antagonists1 item
- HIV3item
- hydroxymethylglutaryl-CoA reductase Inhibitor2item
- Imidazoles1 item
- Immunology/Inflammation49item
- inhibitor1 item
- IP receptor Agonist2item
- Isothiocyanates1 item
- JAK2item
- JAK/STAT Signaling3item
- KCa1.1 Channel blocker2item
- KCa3.1 Channel blocker2item
- Keap1-Nrf22item
- kinase insert domain receptor Inhibitor3item
- kisspeptin receptor Agonist2item
- KNa1.1 Activator3item
- Kv1.2 Channel blocker2item
- Kv1.3 Channel blocker2item
- Kv1.8 Channel blocker2item
- Kv10.1 Channel blocker2item
- Kv11.1 Channel blocker2item
- leucine rich repeat kinase 2 Inhibitor4item
- Liver X receptor-α Antagonist2item
- Liver X receptor-β Antagonist2item
- LPA1 receptor Antagonist2item
- LPA2 receptor Antagonist3item
- LPA3 receptor Antagonist3item
- M1 receptor Antagonist5item
- M2 receptor Antagonist6item
- M3 receptor Antagonist5item
- M4 receptor Antagonist7item
- M5 receptor Antagonist5item
- mAChR2item
- MAPK/ERK Pathway20item
- Material synthetic block1 item
- MC3 receptor Antagonist2item
- MC4 receptor Antagonist2item
- mechanistic target of rapamycin kinase Inhibitor7item
- Membrane Transporter/Ion Channel6item
- Metabolic Enzyme/Protease14item
- mGlu1 receptor Agonist3item
- mGlu1 receptor Allosteric modulator9item
- mGlu1 receptor Antagonist7item
- mGlu2 receptor Agonist2item
- mGlu2 receptor Allosteric modulator2item
- mGlu2 receptor Antagonist3item
- mGlu3 receptor Allosteric modulator3item
- mGlu3 receptor Antagonist3item
- mGlu4 receptor Allosteric modulator5item
- mGlu4 receptor Antagonist3item
- mGlu5 receptor Agonist5item
- mGlu5 receptor Allosteric modulator18item
- mGlu5 receptor Antagonist3item
- mGlu6 receptor Antagonist3item
- mGlu7 receptor Allosteric modulator3item
- mGlu7 receptor Antagonist5item
- mGlu8 receptor Allosteric modulator2item
- mGlu8 receptor Antagonist5item
- mGluR2item
- Mineralocorticoid receptor Agonist2item
- Mineralocorticoid receptor Antagonist3item
- mitogen-activated protein kinase 10 Inhibitor2item
- mitogen-activated protein kinase 11 Inhibitor3item
- mitogen-activated protein kinase 14 Inhibitor6item
- mitogen-activated protein kinase kinase 1 Allosteric modulator2item
- MMP1 Inhibitor2item
- MMP2 Inhibitor2item
- Monoamine oxidase A Inhibitor2item
- Morpholines1 item
- Neuronal NOS Inhibitor4item
- Neuronal Signaling13item
- NF- κ B activation inhibitors1 item
- NF-κB2item
- nicotinic acetylcholine receptor α1 subunit Antagonist2item
- Nitrogen donating ligand1 item
- NK1 receptor Antagonist3item
- NK2 receptor Antagonist2item
- NK3 receptor Antagonist4item
- NO Synthase2item
- Non heterocyclic block1 item
- NOP receptor Agonist2item
- NTS1 receptor Agonist2item
- NTS1 receptor Antagonist2item
- NTS2 receptor Agonist2item
- Opioid Receptor3item
- OT receptor Antagonist5item
- OX1 receptor Antagonist8item
- OX2 receptor Antagonist8item
- oxidative stress3item
- P-glycoprotein2item
- P2X4 Antagonist2item
- P2X7 Antagonist2item
- P2Y1 receptor Allosteric modulator2item
- P2Y1 receptor Antagonist2item
- P2Y12 receptor Antagonist2item
- p38 MAPK18item
- PAC1 receptor Agonist2item
- Peroxisome proliferator-activated receptor-α Agonist6item
- Peroxisome proliferator-activated receptor-γ Agonist4item
- Pharmaceutical ingredients13item
- Pharmacology3item
- phenol1 item
- Phenylpropanoids2item
- Phenylpropanoids Coumarins Phenols Polyphenols2item
- Phenylpropanoids Lignans Phenols Monophenols2item
- phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha Inhibitor7item
- phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit beta Inhibitor5item
- phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta Inhibitor6item
- phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma Inhibitor8item
- phosphodiesterase 3A Inhibitor2item
- phosphodiesterase 4A Inhibitor2item
- Phosphorus compounds1 item
- PI3K/Akt/mTOR33item
- Piperazines2item
- Piperidines1 item
- PKA2item
- platelet derived growth factor receptor beta Inhibitor2item
- Polymer / polymer reagent1 item
- polypeptide1 item
- Potassium Channel3item
- PPAR2item
- Pregnane X receptor Agonist2item
- Progesterone receptor Agonist3item
- PROTAC4item
- PROTACs3item
- Protease inhibitors1 item
- proteasome 20S subunit beta 5 Inhibitor2item
- Protein amino acids1 item
- Protein Tyrosine Kinase/RTK7item
- Pyrazoles1 item
- pyridazines1 item
- Pyrimidines5item
- RAC32item
- Rap guanine nucleotide exchange factor 4 Inhibitor2item
- RAR-related orphan receptor-α Agonist3item
- RAR-related orphan receptor-γ Agonist3item
- Regenerative medicine research reagents4item
- regulator of G-protein signaling 4 Inhibitor3item
- Retinoic acid receptor-α Antagonist3item
- Retinoic acid receptor-β Antagonist2item
- Retinoic acid receptor-γ Agonist2item
- Retinoic acid receptor-γ Antagonist4item
- Retinoid X receptor-α Agonist2item
- Retinoid X receptor-α Antagonist4item
- Retinoid X receptor-β Antagonist2item
- S1P1 receptor Agonist5item
- S1P3 receptor Agonist2item
- S1P4 receptor Agonist2item
- S1P5 receptor Agonist4item
- Salt-inducible Kinase (SIK)3item
- SERT Inhibitor3item
- Seven membered ring compound2item
- Six membered carbocyclic compound2item
- Six-Membered Heterocyclic Compounds16item
- SMO Antagonist6item
- Spectroscopic reagent1 item
- spleen associated tyrosine kinase Inhibitor2item
- SST1 receptor Agonist2item
- SST2 receptor Agonist3item
- SST3 receptor Agonist3item
- SST4 receptor Agonist3item
- SST5 receptor Agonist3item
- Stable isotope2item
- STAT62item
- Stem cell biology2item
- Stem Cell/Wnt6item
- Steroids3item
- TAS2R14 Agonist4item
- TAS2R39 Agonist2item
- terpenes2item
- Terpenoids Triterpenes2item
- Tetracycline antibiotics1 item
- Tetracyclines2item
- TGF-beta/Smad4item
- TGF-β Receptor3item
- Thyroid Hormone Receptor2item
- TP receptor Agonist2item
- TP receptor Antagonist5item
- Triazoles1 item
- Trifluoromethylthio compounds1 item
- TRPA1 Activator4item
- TRPC3 Channel blocker4item
- TRPC4 Channel blocker2item
- TRPC5 Channel blocker4item
- TRPC6 Channel blocker3item
- TRPM2 Channel blocker3item
- TRPM7 Channel blocker2item
- TRPM8 Channel blocker3item
- TRPV1 Activator2item
- TRPV1 Channel blocker2item
- TRPV2 Activator2item
- TRPV4 Activator2item
- ULK4item
- UT receptor Antagonist3item
- V1A receptor Antagonist5item
- V1B receptor Antagonist3item
- V2 receptor Antagonist5item
- Vitamin derivatives1 item
- VPAC1 receptor Agonist2item
- VPAC2 receptor Agonist2item
- Y2 receptor Antagonist2item
- α1A-adrenoceptor Agonist1 item
- α1A-adrenoceptor Antagonist6item
- α1B-adrenoceptor Agonist1 item
- α1B-adrenoceptor Antagonist4item
- α1D-adrenoceptor Agonist1 item
- α1D-adrenoceptor Antagonist3item
- α2A-adrenoceptor Agonist1 item
- α2A-adrenoceptor Antagonist5item
- α2B-adrenoceptor Agonist2item
- α2B-adrenoceptor Antagonist6item
- α2C-adrenoceptor Agonist2item
- α2C-adrenoceptor Antagonist7item
- β1-adrenoceptor Agonist3item
- β1-adrenoceptor Antagonist3item
- β2-adrenoceptor Agonist4item
- β2-adrenoceptor Antagonist1 item
- β3-adrenoceptor Agonist2item
- β3-adrenoceptor Antagonist2item
- δ receptor Agonist3item
- δ receptor Antagonist4item
- κ receptor Agonist3item
- κ receptor Antagonist4item
- μ receptor Agonist2item
- μ receptor Antagonist4item
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Grade
Action Type
- ACTIVATOR21item
- AGONIST177item
- ALLOSTERIC MODULATOR59item
- ANTAGONIST331item
- BLOCKER2item
- CHANNEL BLOCKER18item
- CHELATING AGENT1 item
- GATING INHIBITOR7item
- INHIBITOR178item
- INVERSE AGONIST4item
- MODULATOR5item
- PARTIAL AGONIST2item
- POSITIVE ALLOSTERIC MODULATOR2item
- STABILISER1 item
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