CB2R/FAAH modulator-3 - 99%, high purity , CAS No.2876918-67-9

  • ≥99%
Item Number
C646918
Grouped product items
SKUSizeAvailabilityPrice Qty
C646918-5mg
5mg
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$110.90
C646918-10mg
10mg
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$170.90
C646918-25mg
25mg
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$340.90
C646918-50mg
50mg
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$550.90
C646918-100mg
100mg
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$890.90

Basic Description

Specifications & Purity≥99%
Biochemical and Physiological MechanismsCB2R/FAAH modulator-3 (compound 27) is a dual targeting modulator that acts as a CB2R agonist and FAAH inhibitor. The K i values for CB2R/FAAH modulator-3 are 20.1 and 67.6 nM for CB2R and CB1R, respectively, and the IC 50 value for FAAH is 3.4 μM. CB2R/F
Storage TempStore at -20°C
Shipped InIce chest + Ice pads
Product Description

CB2R/FAAH modulator-3 (compound 27) is a dual targeting modulator that acts as a CB2R agonist and FAAH inhibitor. The K i values for CB2R/FAAH modulator-3 are 20.1 and 67.6 nM for CB2R and CB1R, respectively, and the IC 50 value for FAAH is 3.4 μM. CB2R/FAAH modulator-3 can be used in studies related to cancer , deleterious inflammatory cascades occurring in neurodegenerative diseases, and COVID-19 infection

In Vitro

CB2R/FAAH modulator-3 (compound 27)(10 μM) reduces the production of the pro-inflammatory cytokines TNFα, IFN-γ, IL-1β and IL6 in unstimulated monocytes and macrophages. MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Form:Solid

IC50& Target:CB1 67.6 nM (Ki) CB2 20.1 nM (Ki)

Names and Identifiers

Canonical SMILES O=C(C1=C(OCCCCC)C=CC=C1)N[C@@]2(C3)CC4CC3CC(C4)C2
Molecular Weight 341.49

Certificates

Certificate of Analysis(COA)

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Chemical and Physical Properties

SolubilityDMSO : 50 mg/mL (146.42 mM; Need ultrasonic)

Related Documents

Solution Calculators