Used to characterize GluN2B-containing NMDA receptors
Basic Description
Synonyms
2-Carboxy-3-carboxymethylquinoline
Biochemical and Physiological Mechanisms
For use in conjunction with [3H]-homoquinolinic acid to characterize GluN2B (formally NR2B) containing NMDA receptors; selectively inhibits [3H]-homoquinolinic acid binding to non-NMDA sensitive sites.Please refer toIUPHAR Guide to Pharmacologyfor the mos