CP2 TFA - 97%, high purity , CAS No.C414079

  • ≥97%
Item Number
C414079
Grouped product items
SKUSizeAvailabilityPrice Qty
C414079-5mg
5mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$708.90
C414079-25mg
25mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$2,477.90

Histone Demethylase Inhibitors

View related series
JMJD inhibitor

Basic Description

Specifications & Purity≥97%
Biochemical and Physiological MechanismsCP2 is a cyclic peptide that inhibits the JmjC histone demethylases KDM4 with IC50 values of 42 nM and 29 nM for KDM4A and KDM4C, respectively.
Storage TempStore at -20°C
Shipped InIce chest + Ice pads
Product Description

KDM4C (Cell-free assay); KDM4A (Cell-free assay) 29 nM; 42 nM

In vitro

CP2 uniquely binds in the KDM4A substrate-binding pocket. It binds differently to, but competes with, histone substrates in the active site.

Names and Identifiers

Molecular Weight 2010.15(free basis)

Certificates

Certificate of Analysis(COA)

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4 results found

Lot NumberCertificate TypeDateItem
C2412192Certificate of AnalysisJan 23, 2024 C414079
C2412193Certificate of AnalysisJan 23, 2024 C414079
C2412267Certificate of AnalysisJan 23, 2024 C414079
C2412268Certificate of AnalysisJan 23, 2024 C414079

Chemical and Physical Properties

SolubilitySolubility (25°C) In vitro Water: 100 mg/mL (49.74 mM);    

Related Documents

Solution Calculators