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Cyclobenzaprine hydrochloride - 98%, high purity , Serotonin 2c (5-HT2c) receptor antagonist, CAS No.6202-23-9, Serotonin 2c (5-HT2c) receptor antagonist

  • ≥98%
Item Number
C134704
Grouped product items
SKUSizeAvailabilityPrice Qty
C134704-250mg
250mg
In stock
$31.90
C134704-1g
1g
In stock
$105.90
C134704-5g
5g
In stock
$430.90
C134704-25g
25g
In stock
$1,939.90

Basic Description

SynonymsCyclobenzaprine hydrochloride|6202-23-9|Cyclobenzaprine HCL|Flexeril|Flexiban|Amrix|Cycloflex|Tensodox|Cloben|Cyben|Novo-Cycloprine|3-(5H-dibenzo[a,d][7]annulen-5-ylidene)-N,N-dimethylpropan-1-amine hydrochloride|MK 130 hydrochloride|Cyclobenzaprine (hydr
Specifications & Purity≥98%
Biochemical and Physiological MechanismsCyclobenzaprine Hydrochloride is an inhibitor of the serotonin receptor (SR).Cyclobenzaprine hydrochloride is a type of tricyclic skeletal drug, which is commonly used as a muscle relaxant. It is very effective in treating intractable pain of cervical and
Shipped InNormal
Action TypeANTAGONIST
Mechanism of actionSerotonin 2c (5-HT2c) receptor antagonist
Product Description

Cyclobenzaprine HCl is a skeletal muscle relaxant and a central nervous system (CNS) depressant.
A serotonin receptor inhibitor


Product Application

Cyclobenzaprine hydrochloride has been used to study its effects on the muscles of dystrophin-deficient mdx5Cv mice.

Associated Targets

EHMT2 Tchem Histone-lysine N-methyltransferase EHMT2 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

CBX1 Tbio Chromobox protein homolog 1 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

GMNN Tbio Geminin 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

KMT2A Tchem Histone-lysine N-methyltransferase 2A 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

TRPV1 Tclin Transient receptor potential cation channel subfamily V member 1 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

SLCO1B1 Tchem Solute carrier organic anion transporter family member 1B1 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

SLCO1B3 Tchem Solute carrier organic anion transporter family member 1B3 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

PMP22 Tbio Peripheral myelin protein 22 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

LMNA Tbio Prelamin-A/C 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

MPHOSPH8 Tbio M-phase phosphoprotein 8 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

TDP1 Tchem Tyrosyl-DNA phosphodiesterase 1 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

APEX1 Tchem DNA-(apurinic or apyrimidinic site) lyase 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

KCNH2 Tclin Potassium voltage-gated channel subfamily H member 2 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

IMPA1 Tclin Inositol monophosphatase 1 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

GLP1R Tclin Glucagon-like peptide 1 receptor 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

IDH1 Tclin Isocitrate dehydrogenase [NADP] cytoplasmic 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

Names and Identifiers

Pubchem Sid488182768
Pubchem Sid Urlhttps://pubchem.ncbi.nlm.nih.gov/substance/488182768
IUPAC Name N,N-dimethyl-3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,9,11,13-heptaenylidene)propan-1-amine;hydrochloride
INCHI InChI=1S/C20H21N.ClH/c1-21(2)15-7-12-20-18-10-5-3-8-16(18)13-14-17-9-4-6-11-19(17)20;/h3-6,8-14H,7,15H2,1-2H3;1H
InChi Key VXEAYBOGHINOKW-UHFFFAOYSA-N
Canonical SMILES CN(C)CCC=C1C2=CC=CC=C2C=CC3=CC=CC=C31.Cl
Isomeric SMILES CN(C)CCC=C1C2=CC=CC=C2C=CC3=CC=CC=C31.Cl
WGK Germany 3
RTECS HP0875000
PubChem CID 22576
Molecular Weight 311.85
Reaxy-Rn 6247987

Certificates

Certificate of Analysis(COA)

Enter Lot Number to search for COA:

To view the certificate results,please click on a Lot number.For Lot numbers from past orders,please use our order status section

10 results found

Lot NumberCertificate TypeDateItem
J1631025Certificate of AnalysisFeb 18, 2024 C134704
F2305159Certificate of AnalysisMay 12, 2023 C134704
F2305160Certificate of AnalysisMay 12, 2023 C134704
F2305161Certificate of AnalysisMay 12, 2023 C134704
F2305162Certificate of AnalysisMay 12, 2023 C134704
F2305163Certificate of AnalysisMay 12, 2023 C134704
F2305165Certificate of AnalysisMay 12, 2023 C134704
F2305166Certificate of AnalysisMay 12, 2023 C134704
F2305170Certificate of AnalysisMay 12, 2023 C134704
B2318457Certificate of AnalysisFeb 28, 2023 C134704

Chemical and Physical Properties

SolubilitySoluble in ethanol (50 mg/ml), water (>200 mg/ml), and methanol.
SensitivityMoisture sensitive.
Melt Point(°C)217 °C

Safety and Hazards(GHS)

Pictogram(s) GHS06,   GHS07
Signal Danger
Hazard Statements

H301:Toxic if swallowed

H317:May cause an allergic skin reaction

H312:Harmful in contact with skin

H332:Harmful if inhaled

Precautionary Statements

P261:Avoid breathing dust/fume/gas/mist/vapors/spray.

P280:Wear protective gloves/protective clothing/eye protection/face protection.

P302+P352:IF ON SKIN: wash with plenty of water.

P321:Specific treatment (see ... on this label).

P405:Store locked up.

P501:Dispose of contents/container to ...

P264:Wash hands [and …] thoroughly after handling.

P271:Use only outdoors or in a well-ventilated area.

P270:Do not eat, drink or smoke when using this product.

P304+P340:IF INHALED: Remove person to fresh air and keep comfortable for breathing.

P272:Contaminated work clothing should not be allowed out of the workplace.

P333+P313:IF SKIN irritation or rash occurs: Get medical advice/attention.

P362+P364:Take off contaminated clothing and wash it before reuse.

P330:Rinse mouth.

P301+P316:IF SWALLOWED: Get emergency medical help immediately.

P317:Get emergency medical help.

WGK Germany 3
RTECS HP0875000
Reaxy-Rn 6247987
Merck Index 2713

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