Assay Report Card

Basic Information

ID: ALA1000648

Type: Functional

Description: Antagonist activity at human cloned kappa opioid receptor assessed as inhibition of 50 nM U50488H-stimulated GTPgammaS binding by cell based assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
577.692.652.65
577.692.652.65
593.682.362.36
593.682.362.36
593.682.362.36
593.682.362.36
607.712.662.66
607.712.662.66
595.682.792.79
595.682.792.79
501.591.431.43
462.550.950.95
501.591.431.43
487.561.041.04
636.752.152.15
636.752.152.15
636.752.152.15
636.752.152.15
636.752.152.15
636.752.152.15
636.752.102.10
636.752.152.15