ID: ALA1000648
Type: Functional
Description: Antagonist activity at human cloned kappa opioid receptor assessed as inhibition of 50 nM U50488H-stimulated GTPgammaS binding by cell based assay
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA1000648
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
577.69 | 2.65 | 2.65 |
577.69 | 2.65 | 2.65 |
593.68 | 2.36 | 2.36 |
593.68 | 2.36 | 2.36 |
593.68 | 2.36 | 2.36 |
593.68 | 2.36 | 2.36 |
607.71 | 2.66 | 2.66 |
607.71 | 2.66 | 2.66 |
595.68 | 2.79 | 2.79 |
595.68 | 2.79 | 2.79 |
501.59 | 1.43 | 1.43 |
462.55 | 0.95 | 0.95 |
501.59 | 1.43 | 1.43 |
487.56 | 1.04 | 1.04 |
636.75 | 2.15 | 2.15 |
636.75 | 2.15 | 2.15 |
636.75 | 2.15 | 2.15 |
636.75 | 2.15 | 2.15 |
636.75 | 2.15 | 2.15 |
636.75 | 2.15 | 2.15 |
636.75 | 2.10 | 2.10 |
636.75 | 2.15 | 2.15 |