Assay Report Card

Basic Information

ID: ALA1008221

Type: Binding

Description: Inhibition of human recombinant furin assessed as fluorescent Pyr-RTKR-AMC substrate cleavage

Organism: Homo sapiens

Activity Charts

Bioactivity

Activity Types for Assay ALA1008221

Ki

Total(265)

Compound Summary

Parent Molecular Weight	ALogP	Polar Surface Area
1642.94
1368.62
1438.72
1408.69
1412.68
1353.60
1380.68
1353.61
1353.61
1353.61
1381.62
1381.62
1353.61
1366.65
1408.73
1422.76
1422.76
1406.72
1456.78
1495.81
1440.80
1396.68
1472.78
1410.71
1412.75
1423.70
1437.73
1424.69
1446.74
1437.78
1465.79
1380.68
1422.76
1420.74
1466.77
1438.72
1437.78
1394.71
1422.76
1436.79
1436.79
1420.74
1470.80
1509.84
1454.83
1410.71
1424.73
1426.77
1437.73
1451.76
1438.71
1553.85
1452.74
1460.77
1451.80
1479.82
1440.80
1436.79
1638.96
1599.92
1615.92
1396.67
1451.75
1481.78
1455.74
1396.67
1396.67
1396.67
1396.67
1424.68
1424.68
1382.65
1352.62
1356.61
1297.54
1324.61
1297.54
1297.54
1297.54
1325.55
1325.55
1297.54
1326.58
1271.50
1239.50
1239.50
1212.43
1212.43
1240.44
1268.45
1240.44
1241.47
1154.39
1127.32
1383.64
1328.55
1296.55
1296.55
1269.48
1269.48
1297.49
1325.51
1297.49
1298.53
1211.44
1184.37
1425.72
1370.63
1338.63
1338.63
1311.56
1311.56
1339.57
1367.59
1339.57
1340.61
1253.52
1226.45
1453.73
1423.70
1427.69
1368.62
1395.69
1368.62
1368.62
1368.62
1396.63
1396.63
1397.66
1342.58
1310.58
1310.58
1283.51
1283.51
1311.52
1339.53
1311.52
1312.55
1225.47
1198.40
1509.79
1523.82
1551.88
1565.90
1565.90
1549.86
1581.86
1589.88
1583.94
1539.82
1555.89
1566.85
1580.87
1567.83
1580.92
1608.93
1523.82
1565.90
1563.89
1569.92
1565.90
1580.92
1608.93
1509.79
1481.78
1510.78
1541.86
1553.80
1567.83
1585.89
1495.77
1575.86
1551.88
1566.89
1551.88
1569.92
1552.82
1535.83
1566.85
1594.90
1525.79
1539.82
1537.85
1624.93
1601.89
1509.79
1551.88
1549.86
1595.89
1567.83
1566.89
1594.90
1555.89
1551.88
1591.94
1504.81
1421.73
1409.67
1596.87
1768.03
1810.11
1814.10
1856.18
1658.94
1830.10
1872.18
1810.11
1981.27
2023.35
1421.73
1467.76
1438.76
1439.70
1413.66
1354.59
1381.66
1354.59
1354.59
1354.59
1382.60
1382.60
1354.59
1437.77
1423.74
1395.69
1437.77
1471.79
1407.70
1510.83
1455.81
1411.69
1425.72
1427.76
1487.79
1438.71
1452.74
1439.70
1453.73
1461.75
1452.79
1480.80
1441.78
1437.77
1413.73
1425.67
1457.76
1367.64
1447.73
1423.74
1438.76
1423.74
1441.78
1424.69
1438.72
1466.77
1397.66
1411.69
1409.72
1496.80
1473.76
1381.66
1423.74
1439.70
1486.80
1523.82