Basic Information
ID: ALA1044716
Type: Binding
Description: Inhibition of GST-fused rat recombinant DYRK1A expressed in Escherichia coli assessed as [gamma-33P]ATP incorporation after 10 mins by scintillation counting
Organism: Rattus norvegicus
Activity Charts
Bioactivity
Activity Types for Assay ALA1044716
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 307.26 | 3.10 | 3.10 |
| 322.28 | 4.33 | 4.33 |
| 334.34 | 2.61 | 2.61 |
| 480.07 | 4.09 | 4.09 |
| 292.30 | 2.24 | 2.24 |
| 319.32 | 2.62 | 2.62 |
| 465.06 | 4.09 | 4.09 |
| 386.16 | 3.33 | 3.33 |
| 356.18 | 3.00 | 3.00 |
| 371.19 | 3.00 | 3.00 |
| 413.23 | 3.37 | 3.37 |
| 398.22 | 3.38 | 3.38 |
| 401.18 | 3.32 | 3.32 |
| 386.16 | 3.33 | 3.33 |
| 277.28 | 2.24 | 2.24 |
| 401.18 | 3.32 | 3.32 |