Displacement of [125I]cyanopindolol from human beta 1 adrenergic receptor expressed in CHO cells at 10 uM after 3 to 4 hrs by scintillation counter

Basic Information

ID: ALA1105984

Type: Binding

Description: Displacement of [125I]cyanopindolol from human beta 1 adrenergic receptor expressed in CHO cells at 10 uM after 3 to 4 hrs by scintillation counter

Format: BAO_0000219

Organism: Homo sapiens

Cell type: CHO

Target: Beta-1 adrenergic receptor(ALA213)

Document: ALA1155428

Displacement of [125I]cyanopindolol from human beta 1 adrenergic receptor expressed in CHO cells at 10 uM after 3 to 4 hrs by scintillation counter: 1

Associated Items: Associated Bioactivities Associated Compounds

Activity Charts

Bioactivity

Activity Types for Assay ALA1105984

IC50

Total(59)

Compound Summary

Parent Molecular Weight	ALogP	Polar Surface Area
624.71	6.56	6.56
375.47	3.51	3.51
389.50	3.82	3.82
375.47	3.13	3.13
415.50	3.00	3.00
415.50	3.00	3.00
415.50	2.94	2.94
415.50	2.94	2.94
416.49	2.33	2.33
416.48	3.27	3.27
366.43	1.18	1.18
381.44	0.76	0.76
396.52	2.89	2.89
397.50	2.17	2.17
458.59	4.25	4.25
396.52	2.89	2.89
458.59	4.25	4.25
442.52	2.91	2.91
380.45	1.56	1.56
458.56	2.90	2.90
443.51	2.30	2.30
443.51	2.30	2.30
477.59	2.97	2.97
401.47	3.08	3.08
429.52	3.39	3.39
431.50	3.57	3.57
443.55	3.41	3.41
401.47	2.85	2.85
517.63	5.12	5.12
365.44	1.78	1.78
379.46	2.09	2.09
393.49	2.40	2.40
517.63	5.12	5.12
379.46	2.34	2.34
393.49	2.52	2.52
407.52	2.96	2.96
411.53	2.73	2.73
411.53	2.63	2.63
410.54	3.20	3.20
437.54	4.87	4.87
437.54	4.87	4.87
437.54	4.87	4.87
430.55	3.80	3.80
428.50	2.78	2.78
427.51	3.59	3.59
494.62	5.48	5.48
443.59	5.25	5.25
427.50	4.46	4.46
454.57	4.24	4.24
465.60	4.98	4.98
477.57	4.74	4.74
467.57	4.78	4.78
454.57	4.24	4.24
427.51	3.59	3.59
465.60	4.98	4.98
465.60	4.98	4.98
444.58	4.11	4.11
444.58	4.11	4.11
415.93	2.34	2.34