Assay Report Card

Basic Information

ID: ALA1106185

Type: Binding

Description: Inhibition of AP-1 expressed in HEK293 cells assessed as PMA-stimulated transcriptional activation at 1 uM treated 24 hrs before PMA challenge measured after 20 to 24 hrs by luciferase reporter gene assay

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
465.585.625.62
500.026.276.27
522.635.585.58
543.675.025.02
511.676.346.34
466.575.015.01
479.615.935.93
514.056.586.58
557.705.335.33
525.706.656.65
480.595.325.32
514.056.586.58
536.665.885.88
557.705.335.33
539.736.256.25
480.595.325.32
479.615.935.93
514.056.586.58
536.665.885.88
557.705.335.33
539.736.256.25
480.595.325.32
495.605.635.63
573.705.035.03
496.595.025.02
573.705.035.03
573.705.035.03
501.015.675.67
500.026.276.27
534.476.926.92
557.086.236.23
578.125.675.67
501.015.675.67
507.625.825.82
542.066.476.47
585.715.225.22
508.605.225.22