Basic Information
ID: ALA1119823
Type: Binding
Description: Displacement of [3H]N-cyclobutyl-5-methyl-N-(2-(1-methyl-1H-benzo[d]imidazol-2-ylthio)ethyl)-2-(2H-1,2,3-triazol-2-yl)benzamide from human OX1R expressed in CHO cells after 20 hrs by scintillation counting
Format: BAO_0000219
Organism: Homo sapiens
Cell type: CHO
Target: Orexin receptor 1(ALA5113)
Document: ALA1155457
Displacement of [3H]N-cyclobutyl-5-methyl-N-(2-(1-methyl-1H-benzo[d]imidazol-2-ylthio)ethyl)-2-(2H-1,2,3-triazol-2-yl)benzamide from human OX1R expressed in CHO cells after 20 hrs by scintillation counting: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA1119823
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 413.49 | 2.87 | 2.87 |
| 427.51 | 3.26 | 3.26 |
| 413.49 | 2.95 | 2.95 |
| 431.48 | 3.09 | 3.09 |
| 449.46 | 3.23 | 3.23 |
| 417.52 | 2.68 | 2.68 |
| 416.49 | 3.46 | 3.46 |
| 450.93 | 4.11 | 4.11 |
| 413.49 | 2.95 | 2.95 |