Antagonist activity at human PPARgamma-LBD expressed in CHO-K1 cells co-transfected with GAL4 assessed as inhibition of rosiglitazone-induced lucifera...

Basic Information

ID: ALA1176100

Type: Functional

Description: Antagonist activity at human PPARgamma-LBD expressed in CHO-K1 cells co-transfected with GAL4 assessed as inhibition of rosiglitazone-induced luciferase activity by transactivation assay

Format: BAO_0000219

Organism: Homo sapiens

Cell type: CHO-K1

Target: Peroxisome proliferator-activated receptor gamma(ALA235)

Document: ALA1177724

Antagonist activity at human PPARgamma-LBD expressed in CHO-K1 cells co-transfected with GAL4 assessed as inhibition of rosiglitazone-induced luciferase activity by transactivation assay: 1

Associated Items: Associated Bioactivities Associated Compounds

Activity Charts

Bioactivity

Activity Types for Assay ALA1176100

IC50

Total(1)

Parent Molecular Weight	ALogP	Polar Surface Area
414.58	5.48	5.48

Parent Molecular Weight

ALogP

Polar Surface Area

414.58

5.48

Antagonist activity at human PPARgamma-LBD expressed in CHO-K1 cells co-transfected with GAL4 assessed as inhibition of rosiglitazone-induced lucifera...

Basic Information

Activity Charts

Compound Summary