Inhibition of recombinant HDAC9 assessed as inhibition of (S)-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)-...

Basic Information

ID: ALA1216994

Type: Binding

Description: Inhibition of recombinant HDAC9 assessed as inhibition of (S)-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)-6-(2,2,2-trifluoroacetamido)hexanamide processing by 7-amino-4-methylcoumarin release based FLIPR

Format: BAO_0000357

Target:  Histone deacetylase 9(ALA4145)

Document:  ALA1212811

Inhibition of recombinant HDAC9 assessed as inhibition of (S)-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)-6-(2,2,2-trifluoroacetamido)hexanamide processing by 7-amino-4-methylcoumarin release based FLIPR: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
479.533.643.64
557.651.501.50