Basic Information
ID: ALA1217453
Type: Binding
Description: Inhibition of methyl transferase activity of G9a assessed as inhibition of H3K9 methylation by chemiluminescence based oxygen tunneling assay
Activity Charts
Bioactivity
Activity Types for Assay ALA1217453
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 485.68 | 2.62 | 2.62 |
| 401.51 | 2.38 | 2.38 |
| 387.48 | 1.99 | 1.99 |
| 373.50 | 3.00 | 3.00 |
| 399.54 | 3.53 | 3.53 |
| 357.46 | 2.36 | 2.36 |
| 345.45 | 2.22 | 2.22 |
| 336.82 | 2.81 | 2.81 |
| 359.47 | 2.61 | 2.61 |
| 490.65 | 3.87 | 3.87 |
| 414.55 | 2.30 | 2.30 |
| 400.53 | 1.90 | 1.90 |
| 400.53 | 1.95 | 1.95 |
| 385.51 | 3.14 | 3.14 |
| 331.42 | 1.83 | 1.83 |
| 471.65 | 2.23 | 2.23 |
| 499.70 | 3.01 | 3.01 |
| 513.73 | 3.40 | 3.40 |
| 527.76 | 3.79 | 3.79 |
| 471.65 | 2.27 | 2.27 |
| 513.73 | 3.40 | 3.40 |
| 513.73 | 3.40 | 3.40 |
| 511.72 | 3.15 | 3.15 |
| 525.74 | 3.54 | 3.54 |
| 527.71 | 2.39 | 2.39 |
| 484.69 | 4.10 | 4.10 |
| 486.66 | 3.09 | 3.09 |
| 571.77 | 3.97 | 3.97 |
| 485.68 | 2.79 | 2.79 |
| 499.66 | 2.32 | 2.32 |
| 515.70 | 2.24 | 2.24 |
| 541.74 | 2.78 | 2.78 |
| 528.75 | 2.16 | 2.16 |
| 497.69 | 2.66 | 2.66 |
| 428.58 | 2.32 | 2.32 |
| 415.54 | 2.26 | 2.26 |
| 400.53 | 1.90 | 1.90 |