ID: ALA1249119
Type: Binding
Description: Inhibition of NF-kappaB expressed in HEK293 cells assessed as inhibition of TNF-alpha-induced transcriptional activation treated 24 hrs before TNFalpha challenge by luciferase reporter gene assay
Cell type: HEK293
Bioactivity
Activity Types for Assay ALA1249119
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
382.88 | 4.51 | 4.51 |
479.39 | 6.87 | 6.87 |
541.46 | 8.23 | 8.23 |
468.54 | 5.74 | 5.74 |
537.04 | 7.58 | 7.58 |
440.91 | 5.04 | 5.04 |
444.95 | 5.87 | 5.87 |