Assay Report Card

Basic Information

ID: ALA1273378

Type: Binding

Description: Inhibition of His6x-tagged PRMT1-mediated protein arginine methylation expressed in Escherichia coli BL21 (DE3) assessed as retained fractional activity of enzyme at 100 uM using H4(1-20) and [14C]-AdoMet by scintillation counting

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
433.294.324.32
443.572.542.54
386.485.515.51
409.854.684.68
456.512.042.04
425.524.014.01