Assay Report Card

Basic Information

ID: ALA1292370

Type: Binding

Description: Inhibition of human recombinant SET7/9 in cell free system assessed as monomethylation of histone H3 Lys4 residue after 1 hr in presence of 2 uM AdoMet

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
514.59-1.04-1.04
424.46-2.65-2.65
452.52-1.87-1.87
494.60-0.70-0.70
451.53-0.29-0.29