Basic Information
ID: ALA1647445
Type: Binding
Description: Displacement of [3H]Tiagabine from human recombinant GAT1 expressed in HEK293 cells by equilibrium binding assay
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA1647445
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 335.45 | 4.31 | 4.31 |
| 375.56 | 5.04 | 5.04 |
| 353.44 | 4.44 | 4.44 |
| 369.89 | 4.96 | 4.96 |
| 414.34 | 5.07 | 5.07 |
| 403.44 | 5.32 | 5.32 |
| 349.47 | 4.61 | 4.61 |
| 363.50 | 4.87 | 4.87 |
| 411.55 | 5.97 | 5.97 |
| 365.47 | 4.31 | 4.31 |
| 419.44 | 5.20 | 5.20 |
| 371.43 | 4.58 | 4.58 |
| 367.46 | 4.75 | 4.75 |
| 353.44 | 4.44 | 4.44 |
| 369.89 | 4.96 | 4.96 |
| 414.34 | 5.07 | 5.07 |
| 403.44 | 5.32 | 5.32 |
| 349.47 | 4.61 | 4.61 |
| 363.50 | 4.87 | 4.87 |
| 411.55 | 5.97 | 5.97 |
| 365.47 | 4.31 | 4.31 |
| 419.44 | 5.20 | 5.20 |
| 371.43 | 4.58 | 4.58 |
| 367.46 | 4.75 | 4.75 |
| 363.50 | 4.92 | 4.92 |
| 367.46 | 4.75 | 4.75 |
| 381.49 | 5.01 | 5.01 |
| 371.43 | 4.58 | 4.58 |
| 387.88 | 5.10 | 5.10 |
| 421.43 | 5.46 | 5.46 |
| 367.46 | 4.75 | 4.75 |
| 383.92 | 5.27 | 5.27 |
| 417.47 | 5.63 | 5.63 |
| 379.50 | 4.62 | 4.62 |
| 363.50 | 4.92 | 4.92 |
| 381.49 | 5.01 | 5.01 |
| 387.88 | 5.10 | 5.10 |
| 432.33 | 5.21 | 5.21 |
| 437.43 | 5.34 | 5.34 |
| 383.46 | 4.45 | 4.45 |
| 385.45 | 4.89 | 4.89 |
| 435.46 | 5.77 | 5.77 |
| 393.55 | 5.14 | 5.14 |
| 353.44 | 4.40 | 4.40 |
| 359.51 | 5.34 | 5.34 |
| 377.53 | 4.03 | 4.03 |
| 389.59 | 5.43 | 5.43 |
| 403.61 | 5.82 | 5.82 |
| 373.54 | 4.51 | 4.51 |
| 373.54 | 4.51 | 4.51 |
| 387.57 | 4.90 | 4.90 |
| 387.57 | 4.90 | 4.90 |