ID: ALA1696823
Type: Binding
Description: Inhibition of Saccharomyces cerevisiae MKCDR1h multidrug transporter Cdr1p assessed as concentration required to threefold increase in rate of fluorescence signal relative to absence of inhibitor by fluorescein diacetate based high-throughput screening spectrofluorometric assay
Organism: Saccharomyces cerevisiae
Strain: MKCDR1h
Bioactivity
Activity Types for Assay ALA1696823
INH
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
280.42 | 3.88 | 3.88 |
407.51 | 4.95 | 4.95 |
370.59 | 5.89 | 5.89 |
318.87 | 4.89 | 4.89 |
284.43 | 4.24 | 4.24 |
403.98 | 3.94 | 3.94 |
352.43 | 5.26 | 5.26 |
284.43 | 4.24 | 4.24 |
437.53 | 4.31 | 4.31 |
373.95 | 4.58 | 4.58 |
290.82 | 4.29 | 4.29 |
199.28 | 3.89 | 3.89 |
256.37 | 3.64 | 3.64 |
315.87 | 5.19 | 5.19 |
337.46 | 4.50 | 4.50 |
399.63 | 5.04 | 5.04 |
328.48 | 4.50 | 4.50 |
328.48 | 4.50 | 4.50 |
298.45 | 4.63 | 4.63 |
304.85 | 4.68 | 4.68 |
338.40 | 5.05 | 5.05 |
270.40 | 4.03 | 4.03 |
324.37 | 4.66 | 4.66 |