ID: ALA1771981
Type: Binding
Description: Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assay
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA1771981
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
226.03 | 1.58 | 1.58 |
273.03 | 1.43 | 1.43 |
181.58 | 1.47 | 1.47 |
147.13 | 0.82 | 0.82 |
187.20 | 1.61 | 1.61 |
262.27 | 2.50 | 2.50 |
262.27 | 2.66 | 2.66 |
183.11 | 1.10 | 1.10 |
308.25 | 1.75 | 1.75 |
308.25 | 1.75 | 1.75 |
306.28 | 1.55 | 1.55 |
424.46 | 3.76 | 3.76 |
424.46 | 3.76 | 3.76 |
306.28 | 1.40 | 1.40 |
221.64 | 2.26 | 2.26 |
221.64 | 2.26 | 2.26 |
205.19 | 1.75 | 1.75 |
271.19 | 2.51 | 2.51 |
221.64 | 2.26 | 2.26 |
284.70 | 2.95 | 2.95 |
284.70 | 2.95 | 2.95 |
284.70 | 2.95 | 2.95 |
363.60 | 3.72 | 3.72 |
314.73 | 2.96 | 2.96 |
283.71 | 3.56 | 3.56 |
318.16 | 4.21 | 4.21 |
318.16 | 4.21 | 4.21 |
313.74 | 3.57 | 3.57 |
313.74 | 3.57 | 3.57 |
313.74 | 3.57 | 3.57 |
298.73 | 3.14 | 3.14 |
298.73 | 3.14 | 3.14 |
298.73 | 2.98 | 2.98 |
326.78 | 3.76 | 3.76 |
340.81 | 4.00 | 4.00 |
360.80 | 4.68 | 4.68 |
380.88 | 4.93 | 4.93 |
374.83 | 4.55 | 4.55 |
388.85 | 4.59 | 4.59 |
402.88 | 4.98 | 4.98 |
355.78 | 3.03 | 3.03 |
356.77 | 3.50 | 3.50 |
432.86 | 4.33 | 4.33 |
432.86 | 4.33 | 4.33 |
250.26 | 2.30 | 2.30 |
329.15 | 3.06 | 3.06 |
284.70 | 2.95 | 2.95 |
329.15 | 3.06 | 3.06 |
264.28 | 2.61 | 2.61 |
295.25 | 2.21 | 2.21 |
284.70 | 2.95 | 2.95 |
329.15 | 3.06 | 3.06 |
284.70 | 2.95 | 2.95 |
329.15 | 3.06 | 3.06 |