Assay Report Card

Basic Information

ID: ALA1786052

Type: Functional

Description: Antagonist activity at human TRPV1 E600V mutant expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux at 375 uM for 30 mins before capsaicin challenge measured after 48 hrs by fluorometric analysis

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
817.981.481.48
836.001.001.00