Basic Information
ID: ALA1786689
Type: Functional
Description: Antagonist activity at human TRPV1 E649A mutant expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux at 375 uM for 30 mins before capsaicin challenge measured after 48 hrs by fluorometric analysis
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA1786689
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 817.98 | 1.48 | 1.48 |
| 836.00 | 1.00 | 1.00 |