Assay Report Card

Basic Information

ID: ALA1787846

Type: Binding

Description: Inhibition of catalytic activity of recombinant human IRAP transfected in human HEK-293 cells assessed as cleavage of substrate L-leucine-p-nitroanilide to L-leucine and p-nitroaniline measured every 5 mins for 10 to 50 mins by spectrophotometric analysis

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
774.921.191.19
404.423.383.38
492.622.412.41
536.631.701.70
538.651.921.92
524.621.531.53
466.581.901.90
522.601.311.31
522.601.311.31
536.631.701.70
537.620.460.46
448.571.971.97
448.571.971.97
492.622.412.41
492.622.412.41
492.622.412.41