ID: ALA1787846
Type: Binding
Description: Inhibition of catalytic activity of recombinant human IRAP transfected in human HEK-293 cells assessed as cleavage of substrate L-leucine-p-nitroanilide to L-leucine and p-nitroaniline measured every 5 mins for 10 to 50 mins by spectrophotometric analysis
Organism: Homo sapiens
Cell type: HEK293
Bioactivity
Activity Types for Assay ALA1787846
Ki
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
774.92 | 1.19 | 1.19 |
404.42 | 3.38 | 3.38 |
492.62 | 2.41 | 2.41 |
536.63 | 1.70 | 1.70 |
538.65 | 1.92 | 1.92 |
524.62 | 1.53 | 1.53 |
466.58 | 1.90 | 1.90 |
522.60 | 1.31 | 1.31 |
522.60 | 1.31 | 1.31 |
536.63 | 1.70 | 1.70 |
537.62 | 0.46 | 0.46 |
448.57 | 1.97 | 1.97 |
448.57 | 1.97 | 1.97 |
492.62 | 2.41 | 2.41 |
492.62 | 2.41 | 2.41 |
492.62 | 2.41 | 2.41 |