Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calciu...

Basic Information

ID: ALA1804403

Type: Functional

Description: Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calcium mobilization at 10' -12 to 10'-5 M after 2 mins by fluorometric analysis

Format: BAO_0000219

Organism: Homo sapiens

Cell type: CHO-K1

Target:  Pyroglutamylated RFamide peptide receptor(ALA5852)

Document:  ALA1800022

Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calcium mobilization at 10' -12 to 10'-5 M after 2 mins by fluorometric analysis: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
1905.10
758.88-2.16-2.16
701.83-1.28-1.28
994.07-5.03-5.03
1531.69
1620.74
739.83-4.27-4.27
730.82-2.29-2.29
739.83-4.27-4.27
815.93-3.05-3.05
815.93-3.05-3.05
815.93-3.05-3.05
815.93-3.05-3.05
996.180.700.70
906.06-1.21-1.21
758.88-1.94-1.94