Basic Information
ID: ALA1804404
Type: Functional
Description: Antagonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as inhibition of 26RFa-induced calcium mobilization after 2 mins by fluorometric analysis
Format: BAO_0000219
Organism: Homo sapiens
Cell type: CHO-K1
Target: Pyroglutamylated RFamide peptide receptor(ALA5852)
Document: ALA1800022
Antagonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as inhibition of 26RFa-induced calcium mobilization after 2 mins by fluorometric analysis: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA1804404
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 1905.10 | ||
| 994.07 | -5.03 | -5.03 |
| 1531.69 | ||
| 1620.74 | ||
| 739.83 | -4.27 | -4.27 |
| 730.82 | -2.29 | -2.29 |
| 739.83 | -4.27 | -4.27 |
| 815.93 | -3.05 | -3.05 |
| 815.93 | -3.05 | -3.05 |
| 815.93 | -3.05 | -3.05 |
| 815.93 | -3.05 | -3.05 |
| 996.18 | 0.70 | 0.70 |
| 906.06 | -1.21 | -1.21 |
| 758.88 | -1.94 | -1.94 |