Basic Information
ID: ALA1804405
Type: Functional
Description: Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calcium mobilization after 2 mins by fluorometric analysis
Format: BAO_0000219
Organism: Homo sapiens
Cell type: CHO-K1
Target: Pyroglutamylated RFamide peptide receptor(ALA5852)
Document: ALA1800022
Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calcium mobilization after 2 mins by fluorometric analysis: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA1804405
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 842.01 | -0.99 | -0.99 |
| 842.01 | -0.85 | -0.85 |
| 842.01 | -0.99 | -0.99 |
| 842.01 | -0.99 | -0.99 |
| 827.99 | -1.38 | -1.38 |
| 827.99 | -1.24 | -1.24 |
| 813.96 | -1.63 | -1.63 |
| 882.08 | -0.07 | -0.07 |
| 829.96 | -2.66 | -2.66 |
| 3012.43 | ||
| 900.05 | -1.84 | -1.84 |
| 920.04 | -1.57 | -1.57 |
| 950.07 | -1.08 | -1.08 |
| 978.16 | -0.67 | -0.67 |
| 910.00 | -1.98 | -1.98 |
| 857.03 | -1.64 | -1.64 |
| 952.06 | -1.51 | -1.51 |
| 799.93 | -2.02 | -2.02 |
| 2832.18 | ||
| 2820.17 | ||
| 1121.30 | ||
| 2587.93 | ||
| 1478.73 | ||
| 1535.78 | ||
| 2320.60 | ||
| 2021.27 | ||
| 1649.88 | ||
| 1315.55 | ||
| 1228.47 | ||
| 1072.28 | ||
| 944.11 | -3.43 | -3.43 |
| 815.93 | -3.05 | -3.05 |
| 829.96 | -2.66 | -2.66 |
| 829.96 | -2.66 | -2.66 |
| 739.83 | -4.27 | -4.27 |
| 815.93 | -3.05 | -3.05 |
| 2998.45 | ||
| 982.20 | -0.90 | -0.90 |
| 934.11 | -0.48 | -0.48 |
| 2922.30 | ||
| 2775.13 | ||
| 857.97 | -2.87 | -2.87 |