Basic Information
ID: ALA1815456
Type: Functional
Description: Antagonist activity against human muscle-type alpha1beta1gammadelta nAChR in TE671/RD cells assessed as inhibition of carbamylcholine induced 86Rb+ efflux
Organism: Homo sapiens
Cell type: TE671/RD
Activity Charts
Bioactivity
Activity Types for Assay ALA1815456
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 239.75 | 3.30 | 3.30 |
| 301.43 | 3.51 | 3.51 |
| 313.44 | 3.66 | 3.66 |
| 310.44 | 4.28 | 4.28 |
| 392.93 | 6.04 | 6.04 |
| 408.93 | 5.74 | 5.74 |
| 379.94 | 5.57 | 5.57 |
| 307.82 | 3.39 | 3.39 |
| 293.79 | 3.05 | 3.05 |
| 330.86 | 4.68 | 4.68 |
| 392.93 | 6.04 | 6.04 |
| 307.82 | 3.39 | 3.39 |
| 277.34 | 2.53 | 2.53 |