Assay Report Card

Basic Information

ID: ALA1942548

Type: Binding

Description: Activation of human PKM2 assessed as ATP product formation at 57 nM after 1 hr by luminescent pyruvate kinase-luciferase coupled assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
332.382.442.44
332.382.552.55
316.382.602.60
314.413.603.60
305.362.802.80
279.343.243.24
311.414.264.26
295.793.763.76
291.373.113.11
345.464.214.21
317.372.272.27
318.403.063.06
358.463.403.40
344.443.383.38
318.403.063.06
332.432.932.93
344.443.233.23
330.412.622.62
344.443.013.01