Assay Report Card

Basic Information

ID: ALA1954195

Type: Binding

Description: Binding affinity to proteasome in human HeLa cells assessed as fluorescence at 5 uM pretreated with azido-BODIPY-epoxomicin for 2 hrs followed by 4 hrs of incubation with compound measured post washing by SDS-PAGE-based Western blot analysis

Organism: Homo sapiens

Cell type: HeLa

Subcellular Fraction: Proteasome

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
594.782.042.04
526.681.651.65