Assay Report Card

Basic Information

ID: ALA1959246

Type: Binding

Description: Reversible inhibition of human voltage-gated sodium channel 1.2-mediated current expressed in HEK293 cells at -60 to +10 mV holding poteinitial at 1 to 10 uM after 5 mins measured after drug washout by patch clamp electrophysiology

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
283.803.373.37
283.803.373.37
283.803.373.37