Assay Report Card

Basic Information

ID: ALA2014403

Type: Functional

Description: Agonist activity at human recombinant adenosine receptor-1 expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP production at 10 uM preincubated for 45 mins prior forskolin-induction measured after 15 mins by immunoassay relative to 10 uM CPA

Organism: Homo sapiens

Cell type: CHO

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
308.30-1.84-1.84
281.70-0.03-0.03
321.770.970.97
335.801.361.36
363.852.142.14
377.882.532.53
391.902.922.92
375.861.991.99
375.861.991.99
341.771.161.16
323.781.211.21
351.841.991.99
335.801.211.21
349.821.601.60
375.861.991.99