Basic Information
ID: ALA2020714
Type: Binding
Description: Inhibition of human recombinant autotaxin expressed in insect Sf9 cells using FS-3 as substrate at 1 uM preincubated for 10 mins prior substrate addition measured up to 60 mins by FRET-based analysis
Format: BAO_0000219
Organism: Homo sapiens
Cell type: Sf9
Target: Autotaxin(ALA3691)
Document: ALA2016575
Inhibition of human recombinant autotaxin expressed in insect Sf9 cells using FS-3 as substrate at 1 uM preincubated for 10 mins prior substrate addition measured up to 60 mins by FRET-based analysis: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA2020714
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 436.53 | 5.04 | 5.04 |
| 515.47 | 6.44 | 6.44 |
| 368.41 | 3.57 | 3.57 |
| 396.46 | 4.36 | 4.36 |
| 424.52 | 5.14 | 5.14 |
| 452.57 | 5.92 | 5.92 |
| 450.55 | 5.69 | 5.69 |
| 384.48 | 4.51 | 4.51 |
| 412.53 | 5.29 | 5.29 |
| 440.58 | 6.07 | 6.07 |
| 468.64 | 6.85 | 6.85 |
| 466.62 | 6.63 | 6.63 |