Basic Information
ID: ALA2045986
Type: Binding
Description: Inhibition of FLAG-tagged PHD2 expressed in baculovirus infected insect sf9 cells using biotinyl-DLDLEMLAPYIPMDDDFQL as substrate preincubated with compound for 30 mins measured after 2 hrs by time resolved fluorescence analysis
Cell type: Sf9
Activity Charts
Bioactivity
Activity Types for Assay ALA2045986
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 556.58 | 3.09 | 3.09 |
| 510.56 | 3.08 | 3.08 |
| 511.54 | 3.55 | 3.55 |
| 555.66 | 4.63 | 4.63 |
| 584.66 | 4.62 | 4.62 |
| 584.66 | 4.62 | 4.62 |
| 568.59 | 4.15 | 4.15 |
| 522.57 | 3.35 | 3.35 |
| 538.57 | 3.06 | 3.06 |
| 600.68 | 5.25 | 5.25 |
| 586.66 | 4.95 | 4.95 |
| 605.70 | 4.40 | 4.40 |
| 616.68 | 4.55 | 4.55 |
| 574.65 | 4.74 | 4.74 |
| 574.65 | 4.74 | 4.74 |
| 574.65 | 4.74 | 4.74 |
| 577.67 | 5.17 | 5.17 |
| 559.63 | 4.74 | 4.74 |
| 577.65 | 3.96 | 3.96 |
| 591.67 | 4.22 | 4.22 |
| 605.70 | 4.57 | 4.57 |
| 579.62 | 3.96 | 3.96 |
| 593.64 | 4.27 | 4.27 |
| 579.62 | 3.96 | 3.96 |
| 576.66 | 5.17 | 5.17 |
| 630.63 | 5.88 | 5.88 |
| 576.66 | 5.17 | 5.17 |
| 592.66 | 4.87 | 4.87 |
| 576.66 | 5.17 | 5.17 |
| 548.60 | 4.55 | 4.55 |
| 562.63 | 4.86 | 4.86 |
| 548.60 | 4.55 | 4.55 |
| 562.63 | 4.86 | 4.86 |
| 563.62 | 4.26 | 4.26 |
| 548.60 | 4.55 | 4.55 |
| 562.63 | 4.86 | 4.86 |
| 563.62 | 4.26 | 4.26 |
| 386.50 | 3.50 | 3.50 |
| 496.58 | 5.64 | 5.64 |
| 378.50 | 3.69 | 3.69 |
| 378.50 | 3.69 | 3.69 |
| 372.47 | 3.63 | 3.63 |
| 414.55 | 4.76 | 4.76 |
| 415.54 | 4.15 | 4.15 |
| 423.52 | 4.18 | 4.18 |
| 369.47 | 4.29 | 4.29 |
| 420.52 | 4.84 | 4.84 |
| 424.51 | 3.58 | 3.58 |
| 411.47 | 3.83 | 3.83 |
| 421.50 | 4.24 | 4.24 |
| 421.50 | 4.24 | 4.24 |
| 421.50 | 4.24 | 4.24 |
| 467.53 | 3.73 | 3.73 |
| 336.39 | 2.78 | 2.78 |
| 437.50 | 3.82 | 3.82 |
| 419.51 | 3.48 | 3.48 |
| 434.54 | 5.40 | 5.40 |
| 460.58 | 5.72 | 5.72 |
| 434.54 | 5.15 | 5.15 |
| 460.58 | 5.72 | 5.72 |
| 436.52 | 4.55 | 4.55 |
| 422.53 | 4.79 | 4.79 |
| 373.46 | 3.03 | 3.03 |
| 387.49 | 3.34 | 3.34 |
| 438.54 | 3.82 | 3.82 |
| 400.53 | 4.25 | 4.25 |
| 464.57 | 5.42 | 5.42 |
| 448.57 | 5.30 | 5.30 |
| 459.59 | 6.27 | 6.27 |
| 460.58 | 5.66 | 5.66 |
| 460.58 | 5.66 | 5.66 |
| 538.49 | 7.03 | 7.03 |
| 484.60 | 6.14 | 6.14 |
| 503.60 | 5.97 | 5.97 |
| 460.58 | 5.66 | 5.66 |
| 460.58 | 5.66 | 5.66 |
| 425.53 | 4.60 | 4.60 |
| 411.55 | 5.08 | 5.08 |
| 455.56 | 4.53 | 4.53 |
| 426.52 | 4.15 | 4.15 |
| 470.53 | 3.46 | 3.46 |
| 520.59 | 4.56 | 4.56 |
| 519.61 | 5.17 | 5.17 |
| 520.59 | 4.56 | 4.56 |
| 504.59 | 4.86 | 4.86 |
| 519.61 | 5.17 | 5.17 |
| 520.59 | 4.56 | 4.56 |
| 520.59 | 4.56 | 4.56 |
| 578.63 | 4.17 | 4.17 |
| 564.60 | 4.26 | 4.26 |
| 578.63 | 4.56 | 4.56 |
| 578.63 | 4.56 | 4.56 |
| 578.63 | 4.56 | 4.56 |
| 613.07 | 5.22 | 5.22 |
| 613.07 | 5.22 | 5.22 |
| 596.62 | 4.70 | 4.70 |
| 592.66 | 4.87 | 4.87 |
| 592.66 | 4.87 | 4.87 |
| 526.64 | 4.94 | 4.94 |
| 513.56 | 2.63 | 2.63 |