Assay Report Card

Basic Information

ID: ALA2051182

Type: Binding

Description: Competitive inhibition of [3H]m7-GTP binding to human FLAG-His6 tagged eIF4E expressed in Escherichia coli by scintillation proximity assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
537.21-3.54-3.54
377.25-3.77-3.77
453.35-2.26-2.26
487.79-1.61-1.61
487.79-1.61-1.61
487.79-1.61-1.61
501.82-1.41-1.41
515.85-1.02-1.02
483.37-2.23-2.23
517.82-1.58-1.58
562.27-1.47-1.47
501.36-2.09-2.09
508.38-2.36-2.36
551.37-1.21-1.21
535.81-1.44-1.44
530.82-2.02-2.02
527.81-0.86-0.86
516.830.310.31
561.280.420.42
557.880.220.22
475.832.362.36
489.863.243.24
525.843.793.79
531.944.454.45
503.883.413.41
439.863.263.26