Basic Information
ID: ALA2067498
Type: Functional
Description: Agonist activity at human recombinant adenosine A3 receptor expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP production at 10 uM incubated for 30 mins prior to forskolin-stimulation measured after 15 mins by enzyme immunoassay relative to NECA
Organism: Homo sapiens
Cell type: CHO
Activity Charts
Bioactivity
Activity Types for Assay ALA2067498
Efficacy
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 520.33 | 1.07 | 1.07 |
| 463.33 | 1.77 | 1.77 |
| 653.14 | 5.42 | 5.42 |
| 418.46 | 0.30 | 0.30 |
| 419.45 | -0.31 | -0.31 |
| 436.45 | 0.44 | 0.44 |
| 436.45 | 0.44 | 0.44 |
| 436.45 | 0.44 | 0.44 |
| 452.90 | 0.95 | 0.95 |
| 452.90 | 0.95 | 0.95 |
| 452.90 | 0.95 | 0.95 |
| 497.35 | 1.06 | 1.06 |
| 433.47 | -0.12 | -0.12 |
| 454.44 | 0.57 | 0.57 |
| 454.44 | 0.57 | 0.57 |
| 446.51 | 0.86 | 0.86 |
| 474.57 | 1.59 | 1.59 |
| 460.49 | 0.50 | 0.50 |
| 494.56 | 1.96 | 1.96 |
| 468.52 | 1.45 | 1.45 |
| 518.58 | 2.60 | 2.60 |
| 529.00 | 2.52 | 2.52 |
| 546.99 | 2.66 | 2.66 |
| 563.45 | 3.17 | 3.17 |
| 563.45 | 3.17 | 3.17 |
| 564.98 | 2.80 | 2.80 |
| 544.02 | 2.10 | 2.10 |
| 573.01 | 2.22 | 2.22 |
| 605.10 | 4.19 | 4.19 |
| 653.14 | 5.42 | 5.42 |