Basic Information
ID: ALA2072490
Type: Functional
Description: Antagonist activity at human SST3 receptor expressed in CHO cells assessed as inhibition of forskolin/SS-14-stimulated cAMP accumulation preincubated for 15 mins before SS-14 challenge measured after 1 hr by time-resolved fluorescence analysis
Organism: Homo sapiens
Cell type: CHO
Activity Charts
Bioactivity
Activity Types for Assay ALA2072490
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 396.54 | 6.07 | 6.07 |
| 398.51 | 4.91 | 4.91 |
| 398.51 | 4.91 | 4.91 |
| 384.48 | 4.52 | 4.52 |
| 414.58 | 5.63 | 5.63 |
| 430.58 | 4.64 | 4.64 |
| 446.58 | 4.31 | 4.31 |
| 497.64 | 6.13 | 6.13 |
| 397.53 | 4.49 | 4.49 |
| 439.56 | 4.74 | 4.74 |
| 455.56 | 4.96 | 4.96 |
| 454.58 | 4.54 | 4.54 |