Assay Report Card

Basic Information

ID: ALA2089691

Type: Binding

Description: Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf9 cells assessed as inhibition of pRb Ser780 phosphorylation after 60 mins by TR-FRET assay

Organism: Homo sapiens

Cell type: Sf9

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
482.593.613.61
426.523.783.78
476.584.934.93
477.574.334.33
501.594.814.81
457.583.743.74