Basic Information
ID: ALA2091156
Type: Binding
Description: Inhibition of human recombinant TG2 by fluorescent transamidation assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA2091156
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 226.07 | 2.57 | 2.57 |
| 407.49 | 1.89 | 1.89 |
| 262.13 | 2.33 | 2.33 |
| 228.09 | 2.80 | 2.80 |
| 240.10 | 2.25 | 2.25 |
| 226.07 | 2.57 | 2.57 |
| 226.07 | 2.57 | 2.57 |
| 165.17 | 1.95 | 1.95 |
| 280.35 | 1.60 | 1.60 |
| 225.27 | 1.21 | 1.21 |
| 192.17 | 1.72 | 1.72 |
| 215.17 | 2.83 | 2.83 |
| 147.18 | 1.81 | 1.81 |
| 161.20 | 2.12 | 2.12 |
| 429.50 | 2.45 | 2.45 |
| 391.49 | 1.83 | 1.83 |
| 407.49 | 1.05 | 1.05 |
| 413.47 | 2.35 | 2.35 |
| 409.51 | 2.44 | 2.44 |
| 409.51 | 2.44 | 2.44 |
| 409.51 | 2.44 | 2.44 |
| 423.54 | 2.83 | 2.83 |
| 463.48 | 2.99 | 2.99 |
| 477.51 | 3.38 | 3.38 |
| 429.93 | 2.62 | 2.62 |
| 429.93 | 2.62 | 2.62 |
| 423.50 | 1.57 | 1.57 |
| 427.52 | 1.90 | 1.90 |
| 408.48 | 1.18 | 1.18 |
| 408.48 | 1.78 | 1.78 |
| 411.48 | 1.46 | 1.46 |
| 351.43 | 1.80 | 1.80 |
| 458.54 | 2.91 | 2.91 |
| 472.56 | 2.99 | 2.99 |
| 456.52 | 2.13 | 2.13 |
| 442.50 | 1.74 | 1.74 |
| 514.65 | 3.55 | 3.55 |
| 447.49 | 2.59 | 2.59 |
| 425.51 | 2.06 | 2.06 |
| 409.51 | 2.36 | 2.36 |
| 497.50 | 3.47 | 3.47 |
| 465.48 | 2.73 | 2.73 |
| 447.49 | 2.59 | 2.59 |
| 465.48 | 2.73 | 2.73 |
| 463.94 | 3.11 | 3.11 |
| 497.50 | 3.47 | 3.47 |
| 521.60 | 4.25 | 4.25 |
| 443.53 | 2.76 | 2.76 |
| 479.56 | 3.61 | 3.61 |
| 479.56 | 3.61 | 3.61 |
| 521.60 | 4.25 | 4.25 |
| 521.60 | 4.25 | 4.25 |
| 353.40 | 0.88 | 0.88 |
| 367.43 | 1.27 | 1.27 |
| 407.49 | 2.20 | 2.20 |
| 427.53 | 2.28 | 2.28 |
| 363.44 | 1.05 | 1.05 |
| 460.60 | 2.75 | 2.75 |
| 460.60 | 2.89 | 2.89 |
| 406.51 | 1.72 | 1.72 |
| 442.49 | 1.97 | 1.97 |
| 392.48 | 1.33 | 1.33 |
| 457.60 | 2.86 | 2.86 |
| 372.45 | 1.72 | 1.72 |
| 386.48 | 2.03 | 2.03 |
| 386.48 | 2.03 | 2.03 |
| 440.45 | 2.74 | 2.74 |
| 440.45 | 2.74 | 2.74 |
| 371.46 | 2.32 | 2.32 |
| 439.46 | 3.34 | 3.34 |
| 413.54 | 2.75 | 2.75 |
| 427.57 | 3.14 | 3.14 |
| 396.47 | 1.45 | 1.45 |
| 430.49 | 1.85 | 1.85 |
| 364.43 | 0.45 | 0.45 |
| 458.58 | 2.26 | 2.26 |
| 397.46 | 0.84 | 0.84 |
| 431.47 | 1.24 | 1.24 |
| 459.57 | 1.65 | 1.65 |
| 409.51 | 2.08 | 2.08 |
| 429.50 | 2.45 | 2.45 |
| 594.70 | 4.52 | 4.52 |
| 271.14 | 2.70 | 2.70 |
| 313.32 | 0.53 | 0.53 |
| 413.47 | 2.19 | 2.19 |
| 429.93 | 2.71 | 2.71 |
| 239.27 | 3.60 | 3.60 |
| 177.20 | 1.82 | 1.82 |
| 259.31 | 2.44 | 2.44 |
| 666.78 | -0.13 | -0.13 |
| 395.48 | 2.05 | 2.05 |
| 295.36 | 0.41 | 0.41 |
| 429.50 | 2.45 | 2.45 |
| 429.50 | 2.50 | 2.50 |
| 429.50 | 2.50 | 2.50 |
| 429.50 | 2.50 | 2.50 |
| 429.50 | 2.50 | 2.50 |
| 455.54 | 2.70 | 2.70 |
| 431.51 | 2.70 | 2.70 |
| 407.49 | 2.19 | 2.19 |
| 457.55 | 3.14 | 3.14 |
| 457.55 | 3.14 | 3.14 |
| 443.53 | 2.89 | 2.89 |
| 443.53 | 2.89 | 2.89 |
| 443.53 | 2.84 | 2.84 |
| 439.54 | 2.45 | 2.45 |