Basic Information
ID: ALA2155336
Type: Binding
Description: Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate and [gamma32P]ATP after 30 mins by scintillation counting
Organism: Rattus norvegicus
Activity Charts
Bioactivity
Activity Types for Assay ALA2155336
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 202.24 | 1.82 | 1.82 |
| 201.25 | 2.43 | 2.43 |
| 277.35 | 4.59 | 4.59 |
| 307.38 | 4.60 | 4.60 |
| 337.40 | 4.61 | 4.61 |
| 337.40 | 4.61 | 4.61 |
| 367.43 | 4.61 | 4.61 |
| 321.36 | 4.32 | 4.32 |
| 335.39 | 4.36 | 4.36 |
| 374.24 | 5.49 | 5.49 |
| 338.35 | 4.20 | 4.20 |
| 278.34 | 3.98 | 3.98 |
| 308.37 | 3.99 | 3.99 |
| 338.39 | 4.00 | 4.00 |
| 338.39 | 4.00 | 4.00 |
| 368.42 | 4.01 | 4.01 |
| 322.35 | 3.71 | 3.71 |
| 336.38 | 3.75 | 3.75 |
| 375.23 | 4.88 | 4.88 |
| 339.34 | 3.60 | 3.60 |
| 202.24 | 1.82 | 1.82 |
| 278.34 | 3.98 | 3.98 |
| 308.37 | 3.99 | 3.99 |
| 338.39 | 4.00 | 4.00 |
| 338.39 | 4.00 | 4.00 |
| 368.42 | 4.01 | 4.01 |
| 322.35 | 3.71 | 3.71 |
| 336.38 | 3.75 | 3.75 |
| 375.23 | 4.88 | 4.88 |
| 339.34 | 3.60 | 3.60 |
| 203.23 | 1.22 | 1.22 |
| 279.33 | 3.38 | 3.38 |
| 309.35 | 3.39 | 3.39 |
| 339.38 | 3.40 | 3.40 |
| 339.38 | 3.40 | 3.40 |
| 369.41 | 3.40 | 3.40 |
| 323.34 | 3.11 | 3.11 |
| 337.36 | 3.15 | 3.15 |
| 376.21 | 4.28 | 4.28 |
| 340.32 | 2.99 | 2.99 |