Assay Report Card

Basic Information

ID: ALA2166520

Type: Binding

Description: Potency index, ratio of pEC50 for compound to pEC50 for histamine at human H2R-Gsalphas expressed in Sf9 cells at 0.1 nM to 10 uM by steady state GTPase activity assay

Organism: Homo sapiens

Cell type: Sf9

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
157.240.530.53
546.752.302.30
502.630.470.47
564.792.152.15
578.812.542.54
592.842.932.93
620.893.713.71
677.005.275.27
536.731.531.53
564.792.312.31
648.954.654.65
444.540.120.12
472.600.900.90
500.651.681.68
584.814.024.02
578.812.622.62
345.472.032.03
536.731.371.37