Assay Report Card

Basic Information

ID: ALA2166523

Type: Binding

Description: Potency index, ratio of pEC50 for compound to pEC50 for histamine at guinea pig H2R-Gsalphas expressed in Sf9 cells at 0.1 nM to 10 uM by steady state GTPase activity assay

Organism: Cavia porcellus

Cell type: Sf9

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
157.240.530.53
546.752.302.30
502.630.470.47
564.792.152.15
578.812.542.54
592.842.932.93
620.893.713.71
677.005.275.27
761.167.617.61
536.731.531.53
564.792.312.31
648.954.654.65
733.116.996.99
444.540.120.12
472.600.900.90
500.651.681.68
584.814.024.02
668.986.366.36
578.812.622.62
345.472.032.03
536.731.371.37